Results 41 to 50 of about 7,227 (222)

Synthesis of Some New Enaminoketones, Analogous of Milrinone, 4,Pyrones and Related 4-Pyridones [PDF]

open access: yesIranian Journal of Chemistry & Chemical Engineering, 1996
Synthesis of 4-(N,N- dimethylamino)-3-aryl-3-butene-2-one, ethyl-5-aryl-4-oxo-4H-pyran-2-carboxylate, ethyl-5-aryl-4-pyridones-2-carboxylate and 5-aryl-3-cyano-5-methyl-2-pyridones (aryl=3-thienyl, 2-furyl) are described.
Aziz Shahrisa, Salar Hemmati
doaj  

Modular Chiral N-Heterocyclic Carbene Ligands for the Nickel-Catalyzed Enantioselective C–H Functionalization of Heterocycles

open access: yesCHIMIA, 2020
N-Heterocyclic carbenes (NHCs) are the ligands of choice in a large variety of transformations entailing different transition metals. However, the number and variety of chiral NHCs suitable as stereo-controlling ligands in asymmetric catalysis remains ...
Johannes Diesel, Nicolai Cramer
doaj   +1 more source

Synthesis of Functionalized Bicyclic Pyridones Containing the Dithiocarbamate Group Using Thioazlactones, Diamines, and Nitroketene Dithioacetal

open access: yesSynOpen, 2021
An efficient method for the synthesis of highly substituted bicyclic pyridone derivatives containing the dithiocarbamate group is reported via a one-pot three-component reaction of 2-(alkylthio)thio­azlactones, diamines, and nitroketene dithioacetal in ...
Marziyeh Saeedi   +6 more
doaj   +1 more source

Synthesis of Some Novel Heterocyclic and Schiff Base Derivatives as Antimicrobial Agents

open access: yesMolecules, 2015
Treatment of 2,3-diaryloxirane-2,3-dicarbonitriles 1a–c with different nitrogen nucleophiles, e.g., hydrazine, methyl hydrazine, phenyl hydrazine, hydroxylamine, thiosemicarbazide, and/or 2-amino-5-phenyl-1,3,4-thiadiazole, afforded pyrazole, isoxazole ...
Mohamed E. Azab   +2 more
doaj   +1 more source

Crystal structure of 2,6-dimethyl-4-pyridone hemihydrate

open access: yesActa Crystallographica Section E: Crystallographic Communications, 2015
The title compound (systematic name: 2,6-dimethyl-1H-pyridin-4-one hemihydrate), C7H9NO·0.5H2O, has a single planar molecule in the asymmetric unit with the non-H atoms possessing a mean deviation from planarity of 0.021 Å.
Dalena M. Nguyen   +3 more
doaj   +1 more source

Versatile Synthesis of 3,5-Disubstituted 2-Fluoropyridines and 2-Pyridones

open access: yes, 2016
5-Bromo-2-fluoro-3-pyridylboronic acid (3) was prepared in high yield by ortho-lithiation of 5-bromo-2-fluoropyridine (1), followed by reaction with trimethylborate.
Timothy Gallagher (1261572)   +1 more
core   +1 more source

3-Cyano-4,6-dimethyl-2-pyridone (Guareschi pyridone)

open access: yesActa Crystallographica Section E Structure Reports Online, 2004
In the crystal structure of the title compound, C8H8N2O, the mol­ecules form centrosymmetric dimers via N—H⋯O hydrogen bonds.
Victor B. Rybakov   +3 more
openaire   +1 more source

Diversity-oriented functionalization of 2-pyridones and uracils

open access: yesNature Communications, 2021
Diversity-oriented synthesis of 2-pyridone and uracil derivatives is in urgent need in medicinal chemistry as they are useful pharmacophores. Here the authors show that palladium/norbornene cooperative catalysis enabled dual-functionalization of ...
Yong Shang   +8 more
doaj   +1 more source

Pyridonderivate aus 3-Amino-2H-azirinen und Cyclopropenonen

open access: yesCHIMIA, 1978
Reaction of the 3-dimethylamino-2H-azirines 1a and 1b with diphenylcyclopropenone (2a) in ether or acetonitrile leads to the 2-dimethylamino-5,6-diphenyl-4(3H)-pyridones 3a and 3b in 70 and 80% yield, respectively. The structure of these 1:1-adducts has
Stanislav Chaloupka, Heinz Heimgartner
doaj   +1 more source

Palladium-catalyzed selective oxidative olefination and arylation of 2-pyridones

open access: yes, 2012
Substrate-controlled selective oxidative olefination of N-protected 2-pyridones has been achieved under palladium catalysis. The 5-position selectivity was followed for N-protected simple pyridones.
李兴伟   +4 more
core   +1 more source

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