Human metabolism and pharmacological profiling of protonitazepyne and metonitazepyne, two highly potent nitazenes: prediction of main metabolite activity based on µ-opioid receptor docking simulations. [PDF]
Arch ToxicolBerardinelli D +9 more
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Larger Substituents Enhance Stereospecificity in 1,1-Diazene Nitrogen Extrusion through Attenuation of Dynamic Mismatching. [PDF]
JACS AuWu RK, Zhang SQ, Hong X.
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Intelligent design and synthesis of nucleobase and amino acid-based ligands to inhibit the JAK2 enzyme to treat rheumatoid arthritis. [PDF]
Amino AcidsZarei A, Fatahi A.
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Desymmetrization of <i>meso</i>-Pyrrolidines via Oxoammonium-Catalyzed Enantioselective Hydride Transfer. [PDF]
J Am Chem SocRein J +4 more
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Pyrrolidine dithiocarbamate accelerates early recovery of intestinal microvascular oxygenation in a reversible model of hemorrhagic shock in rats. [PDF]
J Transl MedHof S +11 more
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A novel pyrrolidine-chalcone derivative exhibits synergistic anti-cervical cancer activity by dual-targeting MDM2-p53 axis and ferroptosis pathway. [PDF]
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Stereoelectronic and hydrogen-bonding effects on hydroxyproline conformation. [PDF]
Commun ChemMatsumura F +4 more
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Retraction notice to "Pyrrolidine derivatives as α-amylase and α-glucosidase inhibitors: Design, synthesis, structure-activity relationship (SAR), docking studies and HSA binding" [Heliyon 10 (2024) e39444]. [PDF]
HeliyonBhat AA, Tandon N, Singh I.
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Novel Dihydroisoquinolinone-Amide Compounds as GIPR Agonists for Treating Type 2 Diabetes Mellitus and Obesity. [PDF]
ACS Med Chem LettSabnis RW.
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