Results 11 to 20 of about 4,019 (234)
Molecules, 2021 Ten benzoxazole clubbed 2-pyrrolidinones (11–20) as human monoacylglycerol lipase inhibitors were designed on the criteria fulfilling the structural requirements and on the basis of previously reported inhibitors.
Obaid Afzal +5 more
doaj +1 more source
Molecules, 2020 Thiazole derivatives attract the attention of scientists both in the field of organic synthesis and bioactivity research due to their high biological activity.
Birutė Sapijanskaitė-Banevič +4 more
doaj +1 more source
Archiv der Pharmazie, Volume 356, Issue 1, January 2023., 2023 ZEL‐H16 (1) has been disclosed to be a high‐affinity non‐imidazole H3R (partial) agonist. However, it was found that 1 acts as an inverse agonist for Gαi in various assays. Concise structure–activity relationship studies, molecular pharmacology, and docking were used to shed more light on the properties of 1.
Gábor Wágner +12 more
wiley +1 more source
Kolbe anodic decarboxylation as a green way to access 2-pyrrolidinones [PDF]
, 2020 Nootropic compounds are a group of pharmacologically active pyrrolidones. These molecules, which enhance cognition properties and possess a large prescription field, are particularly interesting synthetic targets for the pharmaceutical industry.
Lam, Kevin
core +1 more source
β-Enamino Esters in Heterocyclic Synthesis: Synthesis of Pyrazolone and Pyridinone Derivatives
Molecules, 2010 An efficient and convenient synthesis of pyrrolidinones and pyridinones utilizing enamino esters as starting material has been described. The structures of the compounds obtained were confirmed by spectral and elemental analyses.
Abdellatif Mohamed Salaheldin +1 more
doaj +1 more source
Catalytic Asymmetric Formal [3+2] Cycloaddition of 2-Isocyanatomalonate Esters and Unsaturated Imines: Synthesis of Highly Substituted Chiral γ‐Lactams [PDF]
, 2017 Unlike their isocyano and isothiocyanato analogues, isocyanato esters remain almost unexplored as formal 1,3-dipoles in asymmetric catalytic reactions. The first asymmetric formal [3+2] cycloaddition involving isocyanato esters and electrophilic alkenes ...
Blay Llinares, Gonzalo +4 more
core +2 more sources
Electrochemical Science Advances, Volume 2, Issue 6, December 2022., 2022 Abstract Reasonable design of the core‐shell structure with a high conductive stable substrate is an effective way to solve the huge volume expansion and low intrinsic conductivity of Si‐based anode materials in Li‐ion batteries (LIBs). In this work, the Hydrangea macrophylla‐like composites (Si@NiO@Ni/C) have been successfully synthesized by staged ...
Kunxiang Yu +4 more
wiley +1 more source
Ultrasound-promoted synthesis of pyrrolidin-2-ones in aqueous medium
Orbital: The Electronic Journal of Chemistry, 2012 Pyrrolidin-2-ones have received considerable attention due to their activity in CNS as nootropic drugs. In parallel, the search for environmentally sustainable processes have been triggered the planning of actions related to organic synthesis.
Márcia Silvana Freire Franco +2 more
doaj +1 more source
Reusing Waste Coffee Grounds as Electrode Materials: Recent Advances and Future Opportunities
Global Challenges, Volume 7, Issue 1, January 2023., 2023 Coffee industry produces more than 8 million tons of waste coffee grounds (WCG) annually. In recent decades, upcycling of WCG‐derived carbon into value‐added electrode materials has attracted growing interests owing to their low cost and high electrochemical properties.
Matthew Pagett +3 more
wiley +1 more source
Radical Cyclization of Trichloroacetamides: Synthesis of Lactams [PDF]
, 2018 Trichloroacetamides can act as radical precursors to synthesize nitrogen-containing heterocycles in a variety of processes, mainly involving atom transfer radical cyclizations (ATRC), mediated by Cu(I) or Ru(II) catalysts, and the hydride reductive ...
Bonjoch i Sesé, Josep +3 more
core +1 more source