Results 121 to 130 of about 18,476 (212)

Synthesis, molecular modeling and NAD(P)H:quinone oxidoreductase 1 inducer activity of novel 2-phenylquinazolin-4-amine derivatives [PDF]

, 2016
Abdelaaty A. Shahat, Albena T. Dinkova-Kostova, Knight JA., Mansour S. Alsaid, Maureen Higgins, Mostafa M. Ghorab, Nehal H. Elghazawy, Nesterova NA, Nesterova NA, Reem K. Arafa, Waris G   +10 more
core   +2 more sources

Discovery of EGT710, an Oral Nonpeptidomimetic Reversible Covalent SARS-CoV-2 Main Protease Inhibitor. [PDF]

J Med Chem
Papillon JPN, Yuan J, Hesse MJ, Zhang L, Robinson RI, Ware NF, Hornak V, Karki RG, Kirrane T, Garland K, Joseph S, Moquin SA, Lakshminarayana SB, Tandeske L, Dovala D, Knapp M, Ornelas E, Fuller D, Ho PI, Xie X, Vulic K, Skolnik SM, Gao J, Zambrowski M, Spiess M, Duca JS, Busby SA, Schirle M, Robinson M, Shi PY, Moser HE, Sarko C, Bradner JE, Diagana TT, Tallarico JA.   +34 more
europepmc   +1 more source

Synthesis of 3-(arylamino) quinazoline-2,4(1H,3H)-dione derivatives via TBHP/I2: Molecular docking, MD simulation, DFT, and pharmacological evaluation as MTH1 inhibitors. [PDF]

PLoS One
Karim MG, Mehrdad M, Gheidari D, Gheidari NZ.   +3 more
europepmc   +1 more source

Discovery of cytotoxic indolo[1,2-<i>c</i>]quinazoline derivatives through scaffold-based design. [PDF]

Beilstein J Org Chem
Khabarov DV, Litvinova VA, Dezhenkova LG, Kaluzhny DN, Tikhomirov AS, Shchekotikhin AE.   +5 more
europepmc   +1 more source

Development of substituted 2-(4-(sulfonyl)piperazin-1-yl)quinazoline molecular hybrids as a new class of antimalarials. [PDF]

RSC Adv
Madhav H, Panda A, Datta D, Shaheen K, Rahman A, Khan AT, Bhattacharjee S, Kumar D, Malhotra P, Hoda N.   +9 more
europepmc   +1 more source

Asymmetric α-amidoalkylation. Synthesis of α-substituted piperidines of high enantiomeric purity [PDF]

, 1987
Kärtner, Annerose, Wanner, Klaus Th.
core   +1 more source

Novel 5-Aryl-[1,2,4]triazoloquinazoline Fluorophores: Synthesis, Comparative Studies of the Optical Properties and ICT-Based Sensing Application. [PDF]

Molecules
Kopotilova AE, Permyakova JV, Starnovskaya ES, Moshkina TN, Novikov AS, Slepukhin PA, Nosova EV.   +6 more
europepmc   +1 more source

Insights into the myosin II inhibitory potency of A-ring-modified (S)-blebbistatin analogs [PDF]

, 2017
Bracke, Marc, Roman, Bart, Stevens, Christian, Van den broecke, Tom, Verhasselt, Sigrid   +4 more
core   +2 more sources

A Trifluoromethyl Quinazoline Compound Regulates the Epithelial-Mesenchymal Transition of Prostatic Hyperplasia Cells by Inhibiting the Secretion of TGF-β1 in Stromal Cells. [PDF]

Curr Issues Mol Biol
Chen L, Zhang D, Yu G, Cheng S, Xu B, Yu J, Liu J, Luo H.   +7 more
europepmc   +1 more source

α_1A-Adrenergic Receptor as a Target for Neurocognition: Cautionary Tale from Nicergoline and Quinazoline Non-Selective Blockers. [PDF]

Pharmaceuticals (Basel)
Perez DM.
europepmc   +1 more source