Results 141 to 150 of about 9,016 (186)
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Quinazoline studies. Part XII. Action of acid and alkali on quinazoline
Journal of the Chemical Society C: Organic, 1968Quinazoline was converted into 2-aminobenzaldehyde and its anhydro-polymers (the trimer, the tetramer, and the monoformyl-tetramer) by the action of hot dilute acid or alkali. The substance of high-molecular weight formed from quinazoline below pH 1·5 was found to be a polymer of the 3,4-adduct of the latter with 2-aminobenzaldehyde.
Adrien Albert, Hiroshi Yamamoto
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5-Substituted quinazoline antifolates
European Journal of Cancer (1965), 1980Abstract Two new 5 -substituted- 2 -amino- 4 -hydroxy-quinazoline antifolates are described. The presence of the 5 -substituent reduced the inhibitory effect upon thymidylate synthetase. In contrast, the 2,4 -diaminoquinazoline series, the same 5 -substituents improved the inhibition.
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Quinazoline Yellow SS in cosmetics
Contact Dermatitis, 1976Five cases of allergic contact dermatitis from Quinazoline Yellow SS (D and C Yellow 11) in cosmetics are described, three from a lipstick and two from a rouge stick. Four of them showed marked oedema spreading to the eyelids and down to the neck. Two of them required systemic steroids.
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1975
Publisher Summary This chapter covers the literature for the period from the latter part of 1994 to the early part of 1998. This period has seen the continued use of pyrimidine drugs—such as AZT and ddC in the treatment of viral diseases and the development of new analogues of these compounds, for example, 3TC (3’-thiocytosine).
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Publisher Summary This chapter covers the literature for the period from the latter part of 1994 to the early part of 1998. This period has seen the continued use of pyrimidine drugs—such as AZT and ddC in the treatment of viral diseases and the development of new analogues of these compounds, for example, 3TC (3’-thiocytosine).
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Quinoline, quinazoline, and acridone alkaloids
Natural Product Reports, 1984The most interesting new alkaloids are the acridones that contain tropone rings, which have been isolated from Citrus species. Emphasis this year is again on synthesis, with highlights including the first use of copper acetylides in the synthesis of furoquinolones, the synthesis of the (1,l -dimethylallyl)quinolinone buchapine, and developments in the ...
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2015
The present invention relates to quinazoline compounds of formula I that function as inhibitors of RET (rearranged during transfection) kinase enzyme activity: (Formula (I)) wherein X, R1, R2, R3, R4, R5, R6 and R7 are each as defined herein. The present invention also relates to processes for the preparation of these compounds, to pharmaceutical ...
Goldberg,, Kristin +7 more
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The present invention relates to quinazoline compounds of formula I that function as inhibitors of RET (rearranged during transfection) kinase enzyme activity: (Formula (I)) wherein X, R1, R2, R3, R4, R5, R6 and R7 are each as defined herein. The present invention also relates to processes for the preparation of these compounds, to pharmaceutical ...
Goldberg,, Kristin +7 more
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