Results 121 to 130 of about 13,731 (218)

RETRACTION: Synthesis, Characterization, and Anticancer Activity of New Quinazoline Derivatives against MCF-7 Cells. [PDF]

ScientificWorldJournal
Journal TSW.
europepmc   +1 more source

From Fragment Hit to Clinical Candidate: Discovery of Dual H1R/H4R Ligands with Superior Efficacy in Allergic Conjunctivitis. [PDF]

J Med Chem
Weber P, Smits R, Lim HD, Andaloussi M, Wijkmans J, de Boer B, Tran TD, Zarzycka B, Dekker ME, van der Meer T, Riemens R, Hauwert N, Wagner G, Vischer HF, Chapin MJ, Gomes P, Whitlock A, Wijtmans M, Leurs R, de Esch IJP.   +19 more
europepmc   +1 more source

Structure-based scaffold hopping reveals strategies to overcome oncogenic KIT and PDGFRA mutation-driven drug-resistance in GIST. [PDF]

Nat Commun
Schulz T, Beerbaum M, Scrima A, Jantzen H, Teuber A, Mühlenberg T, Ebel L, Garcia-Fossa F, George A, Berner N, Weisner J, Müller MP, Wilhelm S, Sievers S, Bauer S, Rauh D.   +15 more
europepmc   +1 more source

Effect of alkyl chain length on the corrosion inhibition performance of 2-thioxo-2,3-dihydroquinazolin-4(1H)-one derivatives for carbon steel in HCl solution. [PDF]

Sci Rep
El-Maksoud SAA, Fathalla W, Saleh MS, El-Dossoki FI.   +3 more
europepmc   +1 more source

New Alkaloids from the Hydrothermal Vent-Derived Fungus <i>Aspergillus clavatus</i> C2WU and Their Mitochondrial Protective and Anti-Photoaging Effects. [PDF]

Mar Drugs
Pan J, Zhou C, Wei J, Simeunovic D, Yan W, Yin Q, Zou M, Wu X, Feng Z, Zhang M, Huang H, Wu B.   +11 more
europepmc   +1 more source

7-Amino-2-(<i>N</i>,<i>N</i>-dimethylamino)quinazoline: a small, bright, easily synthesized scaffold for pH sensors. [PDF]

RSC Adv
Mahdaly M, Maki T, Osako R, Fujimaki Y, Suzuki Y.   +4 more
europepmc   +1 more source

Synthesis and Biological Evaluation of New Quinazolin-4(3H)-One-Coumarin Hybrids Designed as Anticancer and Antibacterial Agents. [PDF]

Int J Mol Sci
Paramonova MP, Novikov MS, Sokhraneva VA, Zhivotova IS, Kezin VA, Zenov MA, Petrushanko IY, Novikova ON, Gorshenin AV, Velikorodnaya YI, Isakova EB, Shchekotikhin AE, Kochetkov SN, Matyugina ES, Khandazhinskaya AL.   +14 more
europepmc   +1 more source

One-Step Synthesis of Dihydropyrroloquinazolinone Alkaloid Natural Products: <i>S</i>‑(-)- and <i>R</i>‑(+)-Vasicinone and Their Novel Analogues. [PDF]

ACS Omega
Khaliq T, Kaur V.
europepmc   +1 more source

In Silico Development of Novel Quinazoline-Based EGFR Inhibitors via 3D-QSAR, Docking, ADMET, and Molecular Dynamics. [PDF]

Int J Mol Sci
Moussaoui M, Baammi S, Baassi M, Kerraj S, Soufi H, Rachdi Y, Idrissi ME, Salah M, Belghiti ME, Daoud R, Belaaouad S.   +10 more
europepmc   +1 more source

Discovery of cytotoxic indolo[1,2-<i>c</i>]quinazoline derivatives through scaffold-based design. [PDF]

Beilstein J Org Chem
Khabarov DV, Litvinova VA, Dezhenkova LG, Kaluzhny DN, Tikhomirov AS, Shchekotikhin AE.   +5 more
europepmc   +1 more source