Results 111 to 120 of about 13,731 (218)

Design, synthesis, and antibacterial activity study of pyrroloquinazoline diamine derivatives. [PDF]

J Enzyme Inhib Med Chem
Cheng M, Tian Y, Shang J, He W, Zheng Y, Yan C, Chen X, Li J, Jiang Y, Fu Q, Deng X, Xiao X, Song M.   +12 more
europepmc   +1 more source

Development of High-Affinity CHD1 Chromodomain Inhibitors. [PDF]

J Med Chem
Greschik H, Friedrich F, Seifert L, Mousavizadeh F, Fiorentino F, Walz J, Zhang L, Li J, Fabbrizi E, Tomassi S, Panahi F, Papenkordt N, Wurnig SL, Osterroth J, Strasser AM, Ruprecht J, Moumbock AFA, Hügle M, Sum M, Peng L, Wang S, Baniahmad AA, Pulido-Cortés L, Timmers HTM, Flaig R, Metzger E, Breit B, Einsle O, Günther S, Rotili D, Mai A, Schüle R, Jung M.   +32 more
europepmc   +1 more source

Quinoline-Based Scaffolds in Anticancer Drug Discovery: Molecular Targets, Synthetic Strategies, and Biological Advances. [PDF]

ChemMedChem
Raza A, Wadhwa P, Sharma S.
europepmc   +1 more source

Synthesis and Antioxidant Properties of Novel Quinazoline Derivatives

Quinazoline derivatives have expressed a broad spectrum of biological activities, but there are few examples in literature on an antioxidant activity of different quinazolines. On the basis of literature by Chinese scientists on the effective antioxidant
Tetere, Zenta, Zicāne, Daina, Rāviņa, Irisa, Rijkure, Inese, Mieriņa, Inese   +4 more
core  

Alkaloids as Emerging Neuroprotective Agents for Neurodegenerative Disorders: Insights into Tryptanthrin and Its Derivatives. [PDF]

Int J Mol Sci
Khan A, Khan H, Park IH, Aldahmash BA, Khan MS, Yang G, Kang KS.   +6 more
europepmc   +1 more source

Ambient and selective synthesis of dihydro-benzimidazoquinazolines in deep eutectic melt of betaine and trichloroacetic acid. [PDF]

RSC Adv
Fadaei Z, Rad-Moghadam K, Pakravan P.
europepmc   +1 more source

Generative AI-Based Drug Design: Target-Aware Molecular Generation for EGFR Type I Inhibitors with Multiplatform Docking Validation. [PDF]

ACS Omega
Khan T, Kwak YB, Kim HC.
europepmc   +1 more source

One-Pot Gateway to Quinazoline-Thiohydantoin Fused Scaffolds and Discovery of Their Antileukemic Activity. [PDF]

JACS Au
Kersting L, Zippel C, Herrmann L, Elbadawi M, Seo EJ, Heckmann F, Saeed MEM, Gaube A, Tailor D, Dheeraj A, Malhotra SV, Muehlich S, Efferth T, Tsogoeva SB.   +13 more
europepmc   +1 more source

Identification of new Trypanosoma cruzi-specific protein synthesis inhibitors by using a developed high-throughput in vitro translation assay. [PDF]

Int J Parasitol Drugs Drug Resist
Mantovani CC, Freitas FRN, Moraes CB, Dos Santos GRR, Cruz LR, Kratz JM, Aktas BH, Schenkman S.   +7 more
europepmc   +1 more source

Design, Synthesis, Antiproliferative Potency and In Silico Studies of Novel Alkynyl Quinazolines as Potential EGFR Inhibitors. [PDF]

Int J Mol Sci
Gkoutzivelaki A, Triantopoulou SI, Chiniadis L, Komiotis A, Triantis C, Komiotis D, Papakyriakou A, Pratsinis H, Manta S.   +8 more
europepmc   +1 more source