Results 101 to 110 of about 9,016 (186)

Gallium/Indium-Promoted [4 + 2] Annulation of 2‑Aminobenzonitriles with Alkynes and Dimerization of 2‑Aminobenzonitriles: One-Pot Access to 4‑Aminoquinolines and 4‑Amino-2-Arylquinazolines. [PDF]

ACS Omega
Sakai N, Ishii M, Yamauchi S, Ogiwara Y, Ishida K.   +4 more
europepmc   +1 more source

Efficient Synthesis and Characterization of Lidocaine Analogue N-Ethyl-N-((8-methylquinazolin-2-yl)methyl)ethanamine

SynOpen
Sang Woo Woo, Jae Ho Shim, Jihye Han, Jin Ju Lim, Hyeon Soo Kim   +4 more
doaj   +1 more source

Quinazolines [<i>a</i>]-Annelated by Five-Membered Heterocycles: Synthesis and Biological Activity. [PDF]

Molecules
Lipunova GN, Nosova EV, Charushin VN.
europepmc   +1 more source

Synthesis of 2-Aryl-4-aminoquinazolines: Design, Molecular Docking, and In Vitro Assessment of Antibacterial and Cytotoxic Potential. [PDF]

Int J Mol Sci
Verdugo F, Braillon C, Mahjoub S, Castro-Alvarez A, Janel-Bintz R, Fechter P, Villa P, Jiménez CA, Donoso-Ruiz DA, Pérez-Fehrmann M, Kesternich V, Ortiz S, Nelson R.   +12 more
europepmc   +1 more source

Design, synthesis, and antimicrobial evaluation of novel quinazoline piperazine phosphorodiamidate hybrids as potent DNA gyrase inhibitors. [PDF]

Sci Rep
Donka SB, Kethineni S, Valaparla BY, Bheemreddy A, Meti MD, More UA, Kotakadi VS, Vatturu M, Doddaga S.   +8 more
europepmc   +1 more source

Multicomponent Synthesis of Multi-Target Quinazolines Modulating Cholinesterase, Oxidative Stress, and Amyloid Aggregation Activities for the Therapy of Alzheimer's Disease. [PDF]

Molecules
Chakhari S, Marco-Contelles J, Iriepa I, Carreiras MDC, Chabchoub F, Ismaili L, Refouvelet B.   +6 more
europepmc   +1 more source

A Series of Pyrazolo-Quinazoline Amines Inhibits the Cytochrome <i>bd</i> Oxidase in <i>Mycobacterium tuberculosis</i>. [PDF]

J Med Chem
Singh S, Ng PS, Lakshmanan U, Mathiyazakan V, Wiggins T, Lee BS, Ang SH, Lin Sim SW, Santos MD, Moraski G, Miller M, Berney M, Grüber G, Pethe K.   +13 more
europepmc   +1 more source

Discovery and Characterization of Divarasib (GDC-6036), a Potent Covalent Inhibitor of KRAS G12C. [PDF]

J Med Chem
Endres NF, Do S, Mroue R, Terrett JA, Saabye M, Oh A, Hunsaker T, Chan E, Tran JC, Nguyen LK, Lian Q, Ma TP, Garner T, Gerosa L, Beresini M, Boudreau A, Bronner SM, Cyr P, Ishisoko N, Izrayelit Y, Jiang F, Kellar T, La H, Labadie S, Lardy M, Liu L, Liu W, Miller S, Rudolph J, Plise E, Sellers BD, Shao C, Wang W, Wang Y, Wei W, Wong S, Yu C, Yu K, Yuen PW, Zang R, Zhang C, Zhou Y, Zhu X, Quinn JG, Ye X, Kiefer JR, Mao J, Evangelista M, Merchant M, Landry ML, Malhotra S, Purkey HE.   +51 more
europepmc   +1 more source

The current status of quinazoline hybrids with antibreast cancer therapeutic potential-part II. [PDF]

Future Med Chem
Zeng H, Zhuang M, Cai F, Lin M, Wang R, Wang J, Zhang H.   +6 more
europepmc   +1 more source