Results 1 to 10 of about 8,749 (208)

One-Pot Gateway to Quinazoline-Thiohydantoin Fused Scaffolds and Discovery of Their Antileukemic Activity. [PDF]

JACS Au
Kersting L, Zippel C, Herrmann L, Elbadawi M, Seo EJ, Heckmann F, Saeed MEM, Gaube A, Tailor D, Dheeraj A, Malhotra SV, Muehlich S, Efferth T, Tsogoeva SB.   +13 more
europepmc   +1 more source

α_1A-Adrenergic Receptor as a Target for Neurocognition: Cautionary Tale from Nicergoline and Quinazoline Non-Selective Blockers. [PDF]

Pharmaceuticals (Basel)
Perez DM.
europepmc   +1 more source

Structure-based scaffold hopping reveals strategies to overcome oncogenic KIT and PDGFRA mutation-driven drug-resistance in GIST. [PDF]

Nat Commun
Schulz T, Beerbaum M, Scrima A, Jantzen H, Teuber A, Mühlenberg T, Ebel L, Garcia-Fossa F, George A, Berner N, Weisner J, Müller MP, Wilhelm S, Sievers S, Bauer S, Rauh D.   +15 more
europepmc   +1 more source

Recent advances in the investigation of the quinazoline nucleus and derivatives with potential anticancer activities. [PDF]

Future Med Chem
Antoniolli G, Lima CSP, Coelho F.
europepmc   +1 more source

A Systematic Review of Synthetic and Anticancer and Antimicrobial Activity of Quinazoline/Quinazolin-4-one Analogues. [PDF]

ChemistryOpen
Manhas N, Kumar G, Dhawan S, Makhanya T, Singh P.   +4 more
europepmc   +1 more source

Potential of Using New Indole- and Benzimidazo[1,2-C]quinazolines in Anticancer Therapy Based on Mesenchymal Stem Cells. [PDF]

Cancer Manag Res
Radzikowska-Bűchner E, Radej S, Niezabitowska E, Sitarz R, Szewc M.   +4 more
europepmc   +1 more source

Antitrypanosomal quinazolines targeting lysyl-tRNA synthetase show partial efficacy in a mouse model of acute Chagas disease. [PDF]

Sci Transl Med
Tulloch LB, Tawell H, Taylor AE, Lima ML, Dawson A, Carvalho S, Wall RJ, Corpas-Lopez V, Dey G, Duggan J, Magalhaes LG, Torrie LS, Frame L, Robinson D, Patterson S, Tinti M, Weaver GW, Robinson WJ, Cal M, Kaiser M, Mäser P, Sjö P, Perry B, Kelly JM, Francisco AF, Bhambra AS, Wyllie S.   +26 more
europepmc   +1 more source

Triple energy transfer-enabled dearomative cycloaddition/rearrangement cascade of bicyclic azaarenes to structurally complex products. [PDF]

Nat Catal
Chahar P, Kundu U, Dutta S, Hölter N, Boser F, Hugel FM, Stadtmann L, Daniliuc CG, Glorius F.   +8 more
europepmc   +1 more source

Does early letermovir initiation delay engraftment? [PDF]

Antimicrob Agents Chemother
Royston L, Gomes CV, Zou M, Van Delden C, Kaiser L, Chalandon Y, Masouridi-Levrat S, Neofytos D.   +7 more
europepmc   +1 more source

Future horizons in diabetes treatment: hypoglycemic activity of [1,2,4]triazino[2,3-<i>c</i>]quinazoline derivatives. [PDF]

Front Endocrinol (Lausanne)
Trzhetsynskyi S, Nosulenko I, Kinichenko A, Skoryna D, Berest H, Shvets V, Voskoboinik O, Kovalenko S, Petakh P, Kamyshnyi O.   +9 more
europepmc   +1 more source