Results 71 to 80 of about 7,050 (179)

Prevention of Weight Regain After GLP1RA Cessation With Oral TIX100

Diabetes, Obesity and Metabolism, Volume 28, Issue 6, Page 5339-5342, June 2026.
SeongHo Jo, Junqin Chen, Gu Jing, Guanlan Xu, Peng Li, Anath Shalev   +5 more
wiley   +1 more source

Facile access to potent antiviral quinazoline heterocycles with fluorescence properties via merging metal-free domino reactions

Nature Communications, 2017
Heterocycles are ubiquitous in bioactive compounds and routes to different substitution patterns are important to access the full substrate space.
Felix E. Held, Anton A. Guryev, Tony Fröhlich, Frank Hampel, Axel Kahnt, Corina Hutterer, Mirjam Steingruber, Hanife Bahsi, Clemens von Bojničić-Kninski, Daniela S. Mattes, Tobias C. Foertsch, Alexander Nesterov-Mueller, Manfred Marschall, Svetlana B. Tsogoeva   +13 more
doaj   +1 more source

Regioselective quinazoline C2 modifications through the azide–tetrazole tautomeric equilibrium

Beilstein Journal of Organic Chemistry
2-Chloro-4-sulfonylquinazolines undergo functional group swap when treated with an azide nucleophile: 1) the azide replaces the sulfonyl group at the C4 position; 2) the intrinsic azide–tetrazole tautomeric equilibrium directs the nucleofugal sulfinate ...
Dāgs Dāvis Līpiņš, Andris Jeminejs, Una Ušacka, Anatoly Mishnev, Māris Turks, Irina Novosjolova   +5 more
doaj   +1 more source

Design, Synthesis, Pharmacological Evaluation of Quinazolin-4(3H)-Ones Bearing Urea Functionality as Potential VEGFR-2 Inhibitors

Drug Design, Development and Therapy
Mohammad M Al-Sanea,1,* Hani M Hafez,2 Ahmed AB Mohamed,3,* Hamed W El-Shafey,4 Abdullah A Elgazar,5 Samar S Tawfik,4 Wafaa A Ewes,4 Shaimaa Hussein,6 Tariq G Alsahli,6 Abdelrahman Hamdi4 1Department of Pharmaceutical Chemistry, College of ...
Al-Sanea MM, Hafez HM, Mohamed AA, El-Shafey HW, Elgazar AA, Tawfik SS, Ewes WA, Hussein S, Alsahli TG, Hamdi A   +9 more
doaj  

Amino-quinazolines [PDF]

Nature, 1945
A. KILLEN MACBETH, HAROLD J. RODDA
openaire   +1 more source

Computational Methods as Screening Toll for Triazole Natural Products Derivatives as Potential β-Tubulin Inhibitors for Fusarium graminearum

Orbital: The Electronic Journal of Chemistry
Phytopathogenic fungi like Fusarium graminearum are the cause of the disease gibberellosis, also known as Fusarium head blight (FHB). This disease shows significant losses in agriculture and effects on global economy. Nevertheless, this condition can be
Larissa de Souza Gasques, Pedro Alves Bezerra Morais, Arlan da Silva Gonçalves , Heberth de Paula   +3 more
doaj   +1 more source

Discovery of cytotoxic indolo[1,2-<i>c</i>]quinazoline derivatives through scaffold-based design. [PDF]

Beilstein J Org Chem
Khabarov DV, Litvinova VA, Dezhenkova LG, Kaluzhny DN, Tikhomirov AS, Shchekotikhin AE.   +5 more
europepmc   +1 more source

2-Azidobenzaldehyde-Enabled Construction of Quinazoline Derivatives: A Review. [PDF]

Int J Mol Sci
Qiu W, Zhan D, Ma X, Zhang X.
europepmc   +1 more source

Novel 5-Aryl-[1,2,4]triazoloquinazoline Fluorophores: Synthesis, Comparative Studies of the Optical Properties and ICT-Based Sensing Application. [PDF]

Molecules
Kopotilova AE, Permyakova JV, Starnovskaya ES, Moshkina TN, Novikov AS, Slepukhin PA, Nosova EV.   +6 more
europepmc   +1 more source

Multicomponent Synthesis of Multi-Target Quinazolines Modulating Cholinesterase, Oxidative Stress, and Amyloid Aggregation Activities for the Therapy of Alzheimer's Disease. [PDF]

Molecules
Chakhari S, Marco-Contelles J, Iriepa I, Carreiras MDC, Chabchoub F, Ismaili L, Refouvelet B.   +6 more
europepmc   +1 more source