Characteristics of muscarinic acetylcholine receptors in rat brain. [PDF]
, 1983 Characteristics of muscarinic acetylcholine (ACh) receptors were studied in the rat central nervous system (CNS) using 3H-quinuclidinyl benzilate (QNB), an antagonist of muscarinic ACh receptors. Scatchard analysis indicated that the rat CNS had a single
Nukina, Itaru
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Expression of functional M2 muscarinic acetylcholine receptor in Escherichia coli [PDF]
, 2000 The M2 muscarinic acetylcholine receptor mutant (M2 mutant), with a lack of glycosylation sites, a deletion in the central part of the third inner loop, and the addition of a six histidine tag at the C-terminus, was fused to maltose binding protein (MBP)
Furukawa, H., Haga, T.
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The Hypoxia Screen as an Indicator of Alterations in the Number of Centeral Cholinergic Recpetors Inuduced by Chronic Acetylcholinestrerase Inhibition [PDF]
, 1982 Chronic administration of diisopropyl fluorophosphate (DFP) at 72 hour intervals for a total of 14 doses resulted in a reduction in the number of central muscarinic receptors in mice as measured by the specific binding of [3H]Quinuclidinyl benzilate (QNB)
Wallace, Kathleen B
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Sequestration of Muscarinic Cholinergic Receptors in Permeabilized Neuroblastoma Cells [PDF]
, 1994 The feasibility of using a permeabilized preparation of human SH-SY-5Y neuroblastoma cells for studies of muscarinic acetylcholine receptor (mAChR) sequestration has been evaluated. Exposure of cells permeabilized with digitonin, streptolysin-O, or the Α-
Fisher, Stephen K. +2 more
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Abstracts of the International Symposium on Dementia in Parkinson’s Disease
, 1994 Behavioural Neurology, Volume 7, Issue 1, Page 5-36, 1994.
wiley +1 more source
Regulation by isoproterenol of muscarinic acetylcholine receptor numbers and sensitivity in rat submandibular, but not lacrimal, glands [PDF]
, 1982 Chronic administration of -isoproterenol, a [beta]-adrenergic agonist, to male Sprague-Dawley rats increased submandibular gland weights by 3 to 4-fold. This increase resulted from a combination of hyperplasia and hypertrophy of secretory cells. Possible
Hootman, Seth R.
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High affinity uptake of L-glutamate and γ-aminobutyric acid in Drosophila melanogaster [PDF]
, 1987 Preparations having properties resembling those of synaptosomes have been isolated from whole fly homogenates of Drosophila melanogaster using ficoll gradient floatation technique.
Acharya, S. R. +3 more
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Drug Repurposing on G Protein-Coupled Receptors Using a Computational Profiling Approach. [PDF]
Front Mol Biosci, 2021 de Felice A, Aureli S, Limongelli V.
europepmc +1 more source
Choline Acetyltransferase and Carnitine Acetyltransferase Activity in Human Spermatozoa During Capacitation [PDF]
, 1997 The regional distribution of ChAT activity in human spermatozoa is altered during in vitro capacitation and it correlates with the fertilizing potential of sperm.
Eccles, Lisa A.
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Hm1 muscarinic cholinergic receptor internalization requires a domain in the third cytoplasmic loop [PDF]
, 1992 Selected regions of the Hm1 muscarinic cholinergic receptor were mutated to analyze the molecular mechanisms of agonist-induced receptor internalization (or sequestration).
Lameh, J. +5 more
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