Acta Chimica SlovenicaNeurosteroids modulate the function of γ-aminobutyric acid type A (GABAA) receptors in the brain. We showed that GABAA receptors modulate neurosteroid interactions with VDAC. GABA enhanced [3H]6-AziP labeling of VDAC in a concentration-dependent manner.
Natalia Akentieva
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Frontiers in PharmacologyIntroductionAlcohol use disorder (AUD) causes significant morbidity and mortality globally. Ethanol’s rewarding and reinforcing effects are attributed to activation of the mesolimbic dopamine system, increasing accumbal dopamine release. While activation
Davide Cadeddu +7 more
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The human GABA <sub>A</sub> receptor α4 subunit variant Ile114Asn linked to epilepsy impairs membrane expression with β3 and δ subunits. [PDF]
MicroPubl BiolWatson DA +4 more
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GABA<sub>A</sub> receptor dysfunction in autism spectrum disorder: molecular mechanisms and therapeutic opportunities. [PDF]
Front PharmacolRagu Varman D +5 more
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GABA<sub>A</sub> Receptor Modulators as Emerging Therapeutic Agents for Depressive Disorders. [PDF]
Drug Des Devel TherGuan BY, Li Y.
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The endogenous cannabinoid system gates plasticity of tonic GABA inhibition. [PDF]
J PhysiolColangeli R, Conti F.
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Direct modulation of human GABA-A α<sub>1</sub>β<sub>2</sub>γ<sub>2</sub> receptors by the endocannabinoid 2-arachidonoylglycerol: implications for cannabinoid-related ligands and limitations for anxiolytic drug development. [PDF]
Front NeurosciMixcoha E +4 more
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Alterations in the Components of the GABA-Glutamate System During ZIKV Infection: A Neuroscience Approach. [PDF]
Int J Mol SciRengifo AC +9 more
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