Results 21 to 30 of about 46,253 (290)
EFSA Journal, 2020 According to Article 12 of Regulation (EC) No 396/2005, EFSA has reviewed the maximum residue levels (MRLs) currently established at European level for the pesticide active substance amisulbrom.
European Food Safety Authority (EFSA) +20 more
doaj +1 more source
Effect of sulfonamide pollution on the growth of manure management candidate Hermetia illucens.
PLoS ONE, 2019 Antibiotics are commonly used in livestock and poultry farming. Residual antibiotics in manure may lead to antibiotic pollution of soil, surface water, and groundwater through land application and run-off rainfall.
Qiao Gao +6 more
doaj +1 more source
Benzamide-4-Sulfonamides Are Effective Human Carbonic Anhydrase I, II, VII, and IX Inhibitors
Metabolites, 2018 A series of benzamides incorporating 4-sulfamoyl moieties were obtained by reacting 4-sulfamoyl benzoic acid with primary and secondary amines and amino acids. These sulfonamides were investigated as inhibitors of the metalloenzyme carbonic anhydrase (CA,
Morteza Abdoli +3 more
doaj +1 more source
Frontiers in Plant Science, 2012 Plant activators are agrochemicals that protect crops from diseases by activating the plant immune system. To isolate lead compounds for use as practical plant activators, we screened 2 different chemical libraries composed of various bioactive ...
Yoshiteru eNoutoshi +4 more
doaj +1 more source
Sulfonamide-Based Inhibitors of Biotin Protein Ligase as New Antibiotic Leads
, 2019 Here, we report the design, synthesis, and evaluation of a series of inhibitors of Staphylococcus aureus BPL (SaBPL), where the central acyl phosphate of the natural intermediate biotinyl-5′-AMP (1) is replaced by a sulfonamide isostere. Acylsulfamide (6)
Jingxian Yu (1332696) +15 more
core +1 more source
Molecules, 2015 A novel series of benzenesulfonamide derivatives containing 4-aminobenzenesul-fonamide and α-amides branched valproic acid or 2,2-dimethylcyclopropanecarboxylic acid moieties were synthesized and screened for their anticonvulsant activities in mice ...
Zhiming Wang +5 more
doaj +1 more source
Molecules, 2020 We have recently reported that N-alkyl and N-acyl naltrindole (NTI) derivatives showed activities for the δ opioid receptor (DOR) ranging widely from full inverse agonists to full agonists.
Chiharu Iwamatsu +7 more
doaj +1 more source
, 2016 A two-drug combination therapy where one drug targets an offending cell and the other targets a resistance mechanism to the first drug is a time-tested, yet underexploited approach to combat or prevent drug resistance.
Caixia Hou (478556) +7 more
core +1 more source
, 2016 The first catalytic dehydrative condensation of the benzylic C–H bonds of toluene and p-xylene with aromatic aldehydes is reported herein. This protocol provides highly atom-economical access to stilbene and p-distyrylbenzene derivatives, whereby water ...
Eri Shibata (3334260) +5 more
core +1 more source
Evolution and Reduction in Sulfonamide Resistance Genes in Aerobic Compost of Pig Manure
AgricultureThis study identified that the absolute abundance of 15 types of antibiotic resistance genes (ARGs) across 21 organic fertilizer samples ranged between 1.15 × 104 and 6.74 × 1010 copies/g, with sulfonamide ARGs and the intI1 gene exhibiting relatively ...
Yihao Huang +5 more
doaj +1 more source