Results 41 to 50 of about 90,509 (255)
Coumarin sulfonamide derivatives: An emerging class of therapeutic agents
Coumarin sulfonamide is a heterocyclic pharmacophore and an important structural motif which is a core and integral part of different therapeutic scaffolds and analogues.
Irfan Ali +7 more
doaj +1 more source
Identification of Small-Molecule Inhibitors against Meso-2, 6-Diaminopimelate Dehydrogenase from Porphyromonas gingivalis [PDF]
Species-specific antimicrobial therapy has the potential to combat the increasing threat of antibiotic resistance and alteration of the human microbiome.
Chen, Weihau +7 more
core +5 more sources
: Sulfonamides are commonly used antibacterials in commercial poultry, contributing toward the development of multidrug-resistant (MDR) phenotypes among Escherichia coli and that has emerged as global concern.
Muhammad Asif Zahoor +7 more
doaj +1 more source
Asymmetric additions to dienes catalysed by a dithiophosphoric acid. [PDF]
Chiral Brønsted acids (proton donors) have been shown to facilitate a broad range of asymmetric chemical transformations under catalytic conditions without requiring additional toxic or expensive metals.
Hamilton, Gregory +4 more
core +2 more sources
Investigation of Some Antibiotic Residue Levels in Honey Produced in Ardahan Province
Beekeeping has been a major agricultural activity since ancient times. The importance of beekeeping is still present in our country, just like in other parts of the world.
Ertan DOĞAN
doaj +1 more source
Crystal structure of N-[(1S,2S)-2-aminocyclohexyl]-2,4,6-trimethylbenzenesulfonamide
The title compound, C15H24N2O2S, was synthesized via a substitution reaction between the enantiopure (1S,2S)-(+)-1,2-diaminocyclohexane and 2,4,6-trimethylbenzene-1-sulfonyl chloride.
Felix N. Ngassa +2 more
doaj +1 more source
Acylsulfonamide safety-catch linker : promise and limitations for solid-phase oligosaccharide synthesis [PDF]
Safety-catch linkers are useful for solid-phase oligosaccharide synthesis as they are orthogonal to many common protective groups. A new acylsulfonamide safety-catch linker was designed, synthesized and employed during glycosylations using an automated ...
Collot, M. +3 more
core +2 more sources
Synthesis and studies of bissydnone sulfonamides based on 4,4’-diaminodiphenyl methane
3,3’-(4,4’-Diphenyl)bissydnonyl methane (5) was synthesized and subjected to chlorosulfonation followed by amination resulted in to formation of 3,3’-(methylenedi-1,4-phenylene)bis[4-{(4-substituted-amino)sulfonyl} sydnone (7a-j).
Shahrukh T. Asundaria, Keshav C. Patel
doaj +1 more source
Gas-phase acidity of sulfonamides: implications for reactivity and prodrug design [PDF]
A computational study at the density functional theory level was performed on bioactive and model sulfonamides with the aim of determining the factors affecting the acidity of the sulfonamido group.
Gomes, JRB, Gomes, P
core +1 more source
In this work, two classes of Carbonic Anhydrase (CA) inhibitors, sulfonamide and coumarin derivatives linked to pyta moiety (2a-b) and their corresponding rhenium complexes (3a-b), were designed.
Yassine Aimene +9 more
doaj +1 more source

