Results 1 to 10 of about 76,467 (269)
Synthesis of Novel Aryl(heteroaryl)sulfonyl Ureas of Possible Biological Interest
The course of reaction of aryl and heteroaryl sulfonamides with diphenylcarbonate (DPC) and 4-dimethylaminopyridine (DMAP) was found to depend on the pKa of the sulfonamide used.
Maria Gdaniec +8 more
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We report herein the synthesis of some beta-D-galactopyranosylamine and beta-lactosylamine amides and sulfonamides. The interactions of these compounds with lectins from the seeds of Erythrina cristagalli (LEC) and Ricinus communis (RCA120) were ...
Anna Paola Butera +9 more
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Sulfonamides and trimethoprim [PDF]
Sulfonamides and trimethoprim are inexpensive and effective antibacterial drugs that have been used extensively. The use of sulfonamides for systemic use has, however, decreased dramatically for several years, mainly because of resistance development in pathogenic bacteria and allergic side effects. Also the clinical efficiency of trimethoprim has been
openaire +2 more sources
Amidine Sulfonamides and Benzene Sulfonamides: Synthesis and Their Biological Evaluation
New amidine and benzene sulfonamide derivatives were developed and structures of the new products were confirmed by elemental and spectral analysis (FT-IR, ESI-MS, 1HNMR, and 13CNMR).
Muhammad Abdul Qadir +4 more
doaj +1 more source
Degradation kinetics of six sulfonamides in hen eggs under simulated cooking temperatures [PDF]
Six sulfonamides, i.e., sulfadiazine, sulfadimethoxine, sulfamerazine, sulfamethazine, sulfamethoxazole and sulfamonomethoxine, were applied to spike whole hen eggs at 0.1 mg kg-1 eggs.
YING-HUA ZHANG, PENG WU, XIN-HUAI ZHAO
doaj
The sulfonamides and their structurally related derivatives, such as the sulfamates and sulfamides, possess the general formula A-SO2NHR, in which the functional group is either directly bound to an aromatic, heterocyclic, aliphatic, or sugar scaffold ...
Claudiu T. Supuran
doaj +1 more source
Deconstructing Protein Binding of Sulfonamides and Sulfonamide Analogues
Sulfonamides are one of the most important pharmacophores in medicinal chemistry and sulfonamide analogs have gained substantial interest in recent years. However, the protein interactions of sulfonamides and especially of their analogs are underexplored.
Patrick L. Purder +9 more
openaire +3 more sources
Gold-catalyzed intermolecular hydroamination of allenes with sulfonamides
A co-catalyst of (PPh3)AuCl/AgOTf for the intermolecular hydroamination of allenes with sulfonamides is shown. The reaction proceeded smoothly under mild conditions for differently substituted allenes giving N-allylic sulfonamides in good yields with ...
Chen Zhang +3 more
doaj +1 more source
Clinical and epidemiological evolution of modern therapy and measles in children
Clinical and epidemiological research on the evolution of measles in children in Leningrad – St. Petersburg from 1927–2014 with an analysis of the effectiveness of treatment of this infection. Divided into three periods of fighting «child plague».
V. N. Timchenko +5 more
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Antibiotics in Raw Meat Samples: Estimation of Dietary Exposure and Risk Assessment
The extensive use of antibiotics in livestock farming poses increased concerns for human health as residues of these substances are present in edible tissues.
Athina Stavroulaki +11 more
doaj +1 more source

