Photoinduced acylations of sulfoximines and transformations of an N-phthalimidoyl sulfoximine
, 2022 Published by RWTH Aachen University ...
Tu, Yongliang
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Iron-catalyzed synthesis of NH sulfoximines and cyclic sulfoximines
, 2018 Published by ...
Yu, Hao
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N-Trifluoromethylthiolated Sulfoximines
Organic Letters, 2015 Air- and moisture-stable N-trifluoromethylthio sulfoximines have been prepared from N-H-sulfoximines via the corresponding N-Br derivatives in excellent yields. The two-step process starts with an easy-to-perform bromination at the sulfoximine nitrogen, followed by a reaction with silver trifluoromethanethiolate.
Christian, Bohnen, Carsten, Bolm
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The Preparation of Aliphatic Fluorinated Sulfoximines
Synthesis, 2003 This work describes the preparation of an aliphatic series of the N-trifluoromethanesulfonyl-S-trifluoromethyl-S-sulfoximine group. The key step of the synthesis is the imination of fluorinated sulfoxides under experimental conditions, which avoid cleavage of the alkyl group.
Magnier, Emmanuel, Wakselman, Claude
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Strain-release driven reactivity of a chiral SuFEx reagent provides stereocontrolled access to sulfinamides, sulfonimidamides, and sulfoximines [PDF]
Nature CommunicationsEfforts aimed at enriching the chemical and structural diversity of small molecules have invigorated synthetic exploration in the last two decades. Spatially defined molecular functionality serves as the foundation to construct unique chemical space to ...
Paresh R. Athawale +4 more
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Synthesis of Sulfoximines and Sulfonimidamides Using Hypervalent Iodine Mediated NH Transfer
Molecules, 2023 The development of NH transfer reactions using hypervalent iodine and simple sources of ammonia has facilitated the synthesis of sulfoximines and sulfonimidamides for applications across the chemical sciences.
Renzo Luisi, James A. Bull
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Synthesis of α-Sulfoximino Tetrazoles via Azido-Ugi Four-Component Reaction
SynOpen, 2022 The sulfoximine-based tetrazoles have been synthesized via azido-Ugi four-component reactions of sulfoximines, isocyanides, aldehydes, and TMS-azide in MeOH at 70 °C in the presence of InCl3.
C. P. Irfana Jesin +2 more
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Synthesis and Preliminary Screening of the Biological Activity of Sulindac Sulfoximine Derivatives
Applied Sciences, 2023 Sulindac is a well-known anti-inflammatory agent, sometimes employed as an adjuvant in antitumor therapy. Due to the recent interest in sulfoximine for its potential chemotherapeutics, we decided to transform sulindac and its methyl ester into the ...
Cosimo Cardellicchio +6 more
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Autocatalytic photoredox Chan-Lam coupling of free diaryl sulfoximines with arylboronic acids
Nature Communications, 2021 N-Arylation of NH-diaryl sulfoximines faces synthetic challenges among reported methods. Here, the authors present a mild copper-catalyzed photoredox dehydrogenative Chan-Lam coupling of free diaryl sulfoximines and arylboronic acids via an auto ...
Cong Wang +8 more
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One-pot synthesis of N-iodo sulfoximines from sulfides [PDF]
, 2021 This is the first report on the synthesis and characterization of N-iodo sulfoximines. The synthesis was designed as a room temperature one-pot cascade reaction from readily available sulfides as starting compounds, converted into sulfoximines by ...
Zupanc, Anže +3 more
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