Results 151 to 160 of about 46,327 (259)

Design, synthesis, and mechanistic evaluation of novel pyrazole/thiazole chalcone hybrids as dual tubulin polymerization and COX-2 inhibitors with potent antiproliferative activity. [PDF]

RSC Adv
Saleem BAA, Qurtam AA, Shalabi AR, Al-Zharani M, Abass KS, Bräse S, Alotaibi G, Alkhammash A.   +7 more
europepmc   +1 more source

Pyrazole-Thiazole Hybrids: Synthesis and Biological Evaluation against <i>Trypanosoma cruzi</i> and <i>Mycobacterium tuberculosis</i>. [PDF]

ACS Omega
Pereira CN, Orlando LMR, de Oliveira EC, Pereira MCS, Carnero CSC, Delgado OJR, Roque-Borda CA, Pavan FR, Dos Santos MS.   +8 more
europepmc   +1 more source

Design, synthesis, and antiproliferative activity of novel thiazole-based derivatives as tubulin polymerization inhibitors targeting the colchicine binding site. [PDF]

RSC Adv
Al-Wahaibi LH, Elshamsy AM, Ali TFS, Youssif BGM, Bräse S, Abdel-Aziz M, El-Koussi NA.   +6 more
europepmc   +1 more source

Discovery of a Novel Coumarin/Thiazole Chalcone Hybrid as a Potent Dual Inhibitor of Tubulin and Carbonic Anhydrases IX & XII with Promising Anti-Proliferative Activity. [PDF]

Molecules
Saleem BAA, Qurtam AA, Ahmed M, Al-Aouadi RFA, Alrikabi AAA, Hetta HF, Bräse S, Alotaibi G, Alkhammash A, Farhan SM.   +9 more
europepmc   +1 more source

Structure elucidation and evaluation of the antimicrobial and antitumor activities of 5-methylthiazole-based Schiff base and its metal chelates. [PDF]

Sci Rep
Wahdan KM, Mandour HSA, El-Ghamry HA, El-Gamil MM, Khedr AM.   +4 more
europepmc   +1 more source

Design, green synthesis, and bioevaluation of 1,3-thiazole-sulfonamide hybrids as antimicrobial and anti-inflammatory agent. [PDF]

Sci Rep
Alrayes AA, Alshammari AQ, Alshammari AQ, Elkanzi NAA, Ali AM.   +4 more
europepmc   +1 more source

Copper catalyzed synthesis of thiazole derivatives from enaminones, amines and CS₂. [PDF]

Sci Rep
Arman A, Nowrouzi N, Abbasi M.
europepmc   +1 more source

Base-Promoted C→N Carbonyl Shift Enables One-Step Access to aza-β-Lactams from α-Heteroaryl-α-amino Esters. [PDF]

Org Lett
Kristek J, Št'astná N, Pospíšil J.
europepmc   +1 more source

Adamantane-thiazole hybrids and related derivatives: synthesis, crystal structures, in vitro antibacterial, antifungal, and anti-proliferative activities. [PDF]

BMC Chem
El-Monaem HSA, El-Ashmawy MB, Abdel-Aziz NI, Blacque O, Habib E, Thamotharan S, El-Emam AA.   +6 more
europepmc   +1 more source

Thiazole as a Promising Scaffold for the Treatment of Schistosomiasis: In Vitro and In Vivo Activity Against Different Developmental Stages of <i>Schistosoma mansoni</i>. [PDF]

Pharmaceuticals (Basel)
Rocha JVRD, França WWM, Machado AL, Cavalcante LAO, Gonçalves MTV, Aguiar TWA, Marques DSC, Nascimento PHDB, Araújo HDA, Filho IJDC, Lima MDCA, Aires AL.   +11 more
europepmc   +1 more source