Results 51 to 60 of about 12,572 (245)
Advanced Intelligent Discovery, EarlyView.This research demonstrates that the combination of domain knowledge–based multiple regression, multi‐objective Bayesian optimization, and generative models is a suitable prediction tool for candidates of high refractive index polymers, even with the constraints in the model trained on limited data. The experimental validation can reproduce the proposed
Takuya Yokoo +3 more
wiley +1 more source
N-Propargylamines: versatile building blocks in the construction of thiazole cores
Beilstein Journal of Organic Chemistry, 2017 Thiazoles and their hydrogenated analogues are not only key structural units in a wide variety of natural products but they also constitute important building blocks in medicinal chemistry.
S. Arshadi +4 more
doaj +1 more source
Nova Biotechnologica et Chimica, 2018 Substituted thiophene-2-carbaldehydes 1a-dwere utilized in the synthesis of symmetrically substituted thiazolo[5,4-d]thiazoles 3a-d. Bis(5,4-d)thiazoles with thiophene core at the termini are the most employed in the chemistry of materials but exhibit ...
Tokárová Zita, Biathová Anna
doaj +1 more source
Thiazole Ring—A Biologically Active Scaffold
Molecules, 2021 Background: Thiazole is a good pharmacophore nucleus due to its various pharmaceutical applications. Its derivatives have a wide range of biological activities such as antioxidant, analgesic, and antimicrobial including antibacterial, antifungal ...
Anthi Petrou +2 more
doaj +1 more source
, 1986 Carbonyl isothiocyanates react with 5-amino-2-furancarboxylates to give the corresponding acylthioureas which cyclize to condensed derivatives related to furo[2,3-d]thiazoles.
Ivan Tóth, Ján Leško, Michal Uher
core +1 more source
Synthesis of Nodulisporic Acid 2‘ ‘-Oxazoles and 2‘ ‘-Thiazoles
, 2016 The semisynthetic conversion of nodulisporic acid A (1) into a set of three heterocyclic side chain derivatives provided compounds, highlighted by 6, with an improved spectrum of ectoparasiticidal activity and pharmacokinetic profile relative to the ...
Richard Berger (1417021) +11 more
core +1 more source
Die Aza‐Büchner–Curtius–Schlotterbeck‐Reaktion: Selektive Bildung Quartärer Kohlenstoffzentren
Angewandte Chemie, EarlyView.Wir stellen die Aza‐Büchner–Curtius–Schlotterbeck‐(ABCS)‐Reaktion vor: eine milde, katalysatorfreie Methode zur Homologierung von Aryliminen. Im Gegensatz zum traditionellen BCS‐Mechanismus durchläuft das Diazo‐Intermediat eine selektive C─C‐Insertion zur Bildung eines quartären Zentrums.
Simon O. Angerer +6 more
wiley +1 more source
Synthesis of New 3-Heteroarylindoles as Potential Anticancer Agents
Molecules, 2016 2-(3-(1H-Indol-3-yl)-5-(p-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)-4-substituted-5-(substituted diazenyl)thiazoles and 2-(1H-indol-3-yl)-9-substituted-4,7-disubstituted pyrido[3,2-e][1,2,4]triazolo[4,3-a]pyrimidin-5(7H)-ones were synthesized via reaction of ...
Abdou O. Abdelhamid +3 more
doaj +1 more source
Molecules, 2021 Rapidly growing antimicrobial resistance among clinically important bacterial and fungal pathogens accounts for high morbidity and mortality worldwide.
Dovilė Malūkaitė +6 more
doaj +1 more source
, 2015 The C–H arylation of (benzo)oxazoles or (benzo)thiazoles with aryltrimethylammonium triflates was carried out via Pd-catalyzed C–H/C–N cleavage.
Jian-Long Tao (1456900) +2 more
core +1 more source