Foram sintetizados novos derivados peptideomiméticos da tiossemicarbazida e da 2-metil-3-tiossemicarbazida visando-se verificar a influência da porção aminoacídica na atividade biológica.
Santos, Luciene María Farías dos +4 more
core
Octahedral [(8-quinolinyl/phenanthridinyl)amine)Ga(III)] complexes, reactivity, affinity for biomolecules, anti-cancer and computational evaluations. [PDF]
Dlamini PC +7 more
europepmc +1 more source
Exploring New Thiosemicarbazide Derivatives Bearing Imidazolidine Ring as Potential Antimicrobial Agents: Design, Synthesis, and Molecular Dynamics Studies. [PDF]
Başoğlu F +4 more
europepmc +1 more source
Facile Cobalt-supported Zeolite 4 A as ecofriendly catalyst to prepare 2-Furyl- hydrazine-1-carbothioamides and 1,2,4 Triazole-3-thiones with anticancer investigation. [PDF]
Farheen A, Awan AN, Hameed A, Alam SF.
europepmc +1 more source
Synthesis of 1,2,4-Triazole-3-Thiol Derivatives from Thiosemicarbazides and Carboxylic Acids Using Polyphosphate Ester. [PDF]
Tretyakov BA +3 more
europepmc +1 more source
Synthesis, molecular modelling, and evaluation of new mono- and bis-isoxazolines as antibacterial agents: <i>in vitro</i> and <i>in silico</i> analysis. [PDF]
Altharawi A +7 more
europepmc +1 more source
In Vitro Antifungal Activity of Thiosemicarbazide Derivatives with a Nitroimidazole Moiety Against <i>Trichophyton</i> spp. Dermatophytes. [PDF]
Andrzejczuk S, Kosikowska U, Wujec M.
europepmc +1 more source
Quinoline-Based Scaffolds in Anticancer Drug Discovery: Molecular Targets, Synthetic Strategies, and Biological Advances. [PDF]
Raza A, Wadhwa P, Sharma S.
europepmc +1 more source
Discovery of a Novel 4,5-Dihydro-1<i>H</i>-pyrazole-1-carbothioamide Derivative with Cytotoxic, Apoptotic, and ABL1 Inhibitory Activities Against Chronic Myeloid Leukemia. [PDF]
Erkan A +3 more
europepmc +1 more source
Synthesis, Characterization, and Antimicrobial Evaluation of Some Novel Hydrazinecarbothioamides. [PDF]
Dincel ED +5 more
europepmc +1 more source

