Results 151 to 160 of about 9,643 (193)

Synthesis of an affinity ligand (‘UPHIT’) for in vivo acylation of the κ‐opioid receptor [PDF]

, 1989
Brian R. de Costa, Linda C. Band, Richard B. Rothman, Arthur E. Jacobson, Victor Bykov, Agu Pert, Kenner C. Rice   +6 more
openalex   +1 more source

LY2444296, a κ-opioid receptor antagonist, selectively reduces alcohol drinking in male and female Wistar rats with a history of alcohol dependence. [PDF]

Sci Rep
Flores-Ramirez FJ, Illenberger JM, Pascasio G, Terenius L, Martin-Fardon R.   +4 more
europepmc   +1 more source

κ‑opioid receptor agonist, U50488H, inhibits pyroptosis through NLRP3 via the Ca²⁺/CaMKII/CREB signaling pathway and improves synaptic plasticity in APP/PS1 mice. [PDF]

Mol Med Rep, 2021
Song X, Cui Z, He J, Yang T, Sun X.
europepmc   +1 more source

κ-Opioid Receptor Is Colocalized in GnRH and KNDy Cells in the Female Ovine and Rat Brain [PDF]

, 2016
Peyton W. Weems, Christine F. Witty, M. Amstalden, Lique M. Coolen, Robert L. Goodman, Michael N. Lehman   +5 more
openalex   +1 more source

κ-Opioid receptor activation attenuates osteoarthritis synovitis by regulating macrophage polarization through the NF-κB pathway. [PDF]

Acta Biochim Biophys Sin (Shanghai)
Shi Y, Tao H, Li X, Zhang L, Li C, Sun W, Chu M, Chen K, Zhu P, Wang Q, Gu C, Wang L, Yang X, Hao Y.   +13 more
europepmc   +1 more source

Enantiomerically Pure Quinoline-Based κ-Opioid Receptor Agonists: Chemoenzymatic Synthesis and Pharmacological Evaluation. [PDF]

ChemMedChem, 2020
Martin B, Schepmann D, Bernal FA, Schmidt TJ, Che T, Loser K, Wünsch B.   +6 more
europepmc   +1 more source

Dynorphin peptides differentially regulate the human κ opioid receptor

, 2007
Yong Chen, Chongguang Chen, Lee‐Yuan Liu‐Chen   +2 more
openalex   +1 more source

Drug design and synthesis of a novel κ opioid receptor agonist with an oxabicyclo[2.2.2]octane skeleton and its pharmacology

, 2009
Hiroshi Nagase, Akio Watanabe, Toru Nemoto, Noriyuki Yamaotsu, Kohei Hayashida, Mayumi Nakajima, Ko Hasebe, Kaoru Nakao, Hidenori Mochizuki, Shuichi Hirono, H. Fujii   +10 more
openalex   +1 more source

Impact of Pharmacological Manipulation of the κ-Opioid Receptor System on Self-grooming and Anhedonic-like Behaviors in Male Mice [PDF]

, 2019
Eduardo R. Butelman, Bryan D. McElroy, Thomas E. Prisinzano, Mary Jeanne Kreek   +3 more
openalex   +1 more source

Changes in Spinal δ and κ Opioid Systems in Mice Deficient in the A_2AReceptor Gene [PDF]

, 2002
Alexis Bailey, Catherine Ledent, Mary Kelly, Susanna M.O. Hourani, Ian Kitchen   +4 more
openalex   +1 more source