Results 151 to 160 of about 18,261 (204)

Synthesis, Computational Study, and In Vitro α-Glucosidase Inhibitory Action of 1,3,4-Thiadiazole Derivatives of 3-Aminopyridin-2(1H)-ones. [PDF]

Pharmaceuticals (Basel)
Shulgau Z, Palamarchuk IV, Sergazy S, Urazbayeva A, Ramankulov Y, Kulakov IV.   +5 more
europepmc   +1 more source

Synthesis of novel piperazine-based bis(thiazole)(1,3,4-thiadiazole) hybrids as anti-cancer agents through caspase-dependent apoptosis. [PDF]

RSC Adv
Mohamed DM, Kheder NA, Sharaky M, Nafie MS, Dawood KM, Abbas AA.   +5 more
europepmc   +1 more source

Identification of Benzothiazoles Bearing 1,3,4-Thiadiazole as Antiproliferative Hybrids Targeting VEGFR-2 and BRAF Kinase: Design, Synthesis, BIO Evaluation and In Silico Study. [PDF]

Molecules
Ewes WA, Tawfik SS, Almatary AM, Ahmad Bhat M, El-Shafey HW, Mohamed AAB, Haikal A, El-Magd MA, Elgazar AA, Balaha M, Hamdi A.   +10 more
europepmc   +1 more source

Novel quinazolines bearing 1,3,4-thiadiazole-aryl urea derivative as anticancer agents: design, synthesis, molecular docking, DFT and bioactivity evaluations. [PDF]

BMC Chem
Masoudinia S, Samadizadeh M, Safavi M, Bijanzadeh HR, Foroumadi A.   +4 more
europepmc   +1 more source

Some of the next articles are maybe not open access.

Related searches:

1,3,4-Thiadiazole Based Anticancer Agents

Anti-Cancer Agents in Medicinal Chemistry, 2016
In recent years, researchers like medicinal chemists in the field of medicinal chemistry have widely utilized the 1,3,4-thiadiazole nucleus to investigate its biological and pharmacological effects. This heterocyclic structure has demonstrated various bioactivities such as antifungal, antimicrobial, antiviral, antileishmanial, anti-inflammatory ...
Alireza Aliabadi
exaly   +3 more sources

Antiviral 1,3,4-Thiadiazoles

Chemotherapy, 2009
Nine 1,3,4-thiadiazoles showed an antiviral action against Mengo virus; four of them were also active against vaccinia virus and one against fowl plague virus. Investigations with Mengo virus revealed plaque reduction, inhibition of the cytopathic effect and depression of virus multiplication, with the maximum activity after substance addition from 0–2
Marion Tonew, Elke Klimke
openaire   +2 more sources

Solid-Phase Synthesis of 1,3,4-Thiadiazole Derivatives via Desulfurative Cyclization of Thiosemicarbazide Intermediate Resin

ACS Combinatorial Science, 2016
A 1,3,4-thiadiazole library was constructed by solid-phase organic synthesis. The key step of this solid-phase synthesis involves the preparation of polymer-bound 2-amido-5-amino-1,3,4-thiadiazole resin by the cyclization of thiosemicarbazide resin using
Young-Dae Gong, Seung-Ju Yang
exaly   +2 more sources

Microwave spectra of 1,3,4-thiadiazole and [34S]1,3,4-thiadiazole. Dipole moment of 1,3,4-thiadiazole

Journal of Molecular Spectroscopy, 1962
Abstract The microwave spectra of 1, 3, 4-thiadiazole (I) and [ 34 S] 1, 3, 4-thiadiazole (II) have been recorded in the 15,000–30,000 Mc/sec region. Twelve and ten transitions, respectively, were assigned. The rotational constants of (I) are, A = 8907.51 ± 0.10, B = 5569.27 ± 0.02, and C = 3424.80 ± 0.03 Mc/sec. For (II), A = 8908.15 ± 0.20,
Børge Bak, Daniel Christensen, Lise Hansen-Nygaard, Leif Lipschitz, John Rastrup-Andersen   +4 more
openaire   +1 more source

Synthesis and antifungal activity of thiadiazole-functionalized chitosan derivatives

Carbohydrate Research, 2013
A groups of novel water soluble chitosan derivatives containing 1,3,4-thiadiazole group were synthesized including 1,3,4-thiadiazole (TPCTS), 2-methyl-1,3,4-thiadiazole (MTPCTS), and 2-phenyl-1,3,4-thiadiazole (PTPCTS).
Qing Li, Zhanyong Guo, Guodong Gu
exaly   +2 more sources

Synthesis of 1,3,4-thiadiazole oligomers

Journal of the Chemical Society, Perkin Transactions 1, 2002
AbstractFor Abstract see ChemInform Abstract in Full Text.
Van‐Duc Le, Charles W. Rees, Sivaprasad Sivadasan   +2 more
openaire   +1 more source