Results 51 to 60 of about 43,455 (160)
Aktualʹnì Pitannâ Farmacevtičnoï ì Medičnoï Nauki ta Praktiki, 2017 Introduction. Heterocyclic system of 1,2,4-triazole is interesting and has a popularity among scientists around the world every year. Most attention today is attracted to the compounds formed by a combination of 1,2,4-triazole and various structural ...
D. M. Danilchenko +2 more
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Antidepressant Activity of Some Novel 1, 2, 4 Triazole Substituted Quinazoline Derivatives
International Journal of Pharmaceutical Chemistry and Analysis, 2016 Introduction: Quinazoline is an important moiety found natural and used for their biological activity, quinazoline always attract scientist due to its broad therapeutic value. In the present research article we prepared a series of fifteen compound by conjugating to prominent therapeutic active moiety to produce synergistic effect to mimic the ...
Narendra Joshi, Anju Goyal
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Química NovaEugenol is an aromatic compound found in several plant species. It presents important biological activities including cytotoxicity. In this paper, it is described the synthesis and the evaluation of the cytotoxic activity of eugenol derivatives bearing 1,
Poliana Aparecida Rodrigues Gazolla +8 more
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Aktualʹnì Pitannâ Farmacevtičnoï ì Medičnoï Nauki ta Praktiki, 2016 The aim of this work was the synthesis of new highly effective and low-toxic substances in a series of 5-(quinoline-2-yl, 2-hydroxyquinoline-4-yl)-4-R1-2,4-dyhydro-3Н-1,2,4-triazole-3-thiones and its derivatives, and also establishment of physical ...
T. M. Kaplaushenko
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Chemical Structure and Herbicidal Activity of 1, 2, 4-Triazole-carboxamide Derivatives.
Journal of Weed Science and Technology, 1999 新規な1,2,4-トリアゾールカルボキサミド誘導体について, タイヌビエに対する除草活性と移植イネに対する安全性を指標として, 構造と活性を検討した。1. 雑草発生前処理高いタイヌビエ除草活性と移植イネに対する安全性を保有するには, ベンゼン環の2位と6位が低級アルキル基や塩素原子で置換されていることが必要で, とくに2,6-ジメチル置換体, 2-メチル-6-エチル置換体, 2-メチル-6-塩素置換体および2,4,6-トリメチル置換体が, 優れた除草活性とイネ安全性を示した。カルバモイル基の置換様式は, N,N-ジエチルカルバモイル体およびN-エチル, N-プロピカルバモイル体が高活性に寄与し, アルキル基がメチルあるいはブチルでは劣った。イネに対してはいずれも高い安全性を示した ...
Mitsuru Kanzaki +2 more
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International Journal of Electrochemical Science, 2012 The corrosion inhibition properties of three triazoles derivatives namely 4-amino-5-phenyl-4H-1, 2, 4,-triazole-3-thiol (APTT), 4-amino-5-(2-hydroxy) phenyl-4H-1, 2, 4,-triazole-3-thiol, (AHPTT), 4-amino-5-styryl-4H-1, 2, 4,-triazole-3-thiol, (ASTT) on ...
M.A. Quraishi +3 more
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Analgesic activity of 4-amino-5-methyl-4H-1,2,4-triazol-3-thiones
Aktualʹnì Pitannâ Farmacevtičnoï ì Medičnoï Nauki ta Praktiki, 2018 Аbstract Significance. Nowadays non-steroidal anti-inflammatory drugs have found a wide application in treatment of medical conditions. Despite the clinical effectiveness of non-steroidal anti-inflammatory drugs, their administration is followed by a ...
T. V. Kravchenko +2 more
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Synthesis of substituted 1, 2, 4-triazole derivatives by Microwave irradiation
IOSR Journal of Applied Chemistry, 2013 Various substituted Triazole-Thiol containing different functional group have been synthesized by microwave method. The title product 1-((3H-indol-2-ylamino) methyl)-4-phenyl-4, 5-dihydro-1H-1, 2, 4- triazole-3-thiol is synthesized by using amino benzothiazole.
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Aktualʹnì Pitannâ Farmacevtičnoï ì Medičnoï Nauki ta PraktikiThis study presents the computational prediction of acute toxicity for new derivatives of 3,5-bis(5-mercapto-4-R-4H-1,2,4-triazol-3-yl)phenols and their alkylated analogues.
K. K. Isaicheva, A. H. Kaplaushenko
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Aktualʹnì Pitannâ Farmacevtičnoï ì Medičnoï Nauki ta PraktikiThe activation of lipid free radical oxidation is a key stage in the development of many diseases and can lead to the emergence of related complications.
I. M. Bilai +4 more
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