A REVIEW: THIAZINES DERIVATIVES TREATED AS POTENTIAL ANTIMICROBIAL AGENTS [PDF]
, 2017 In recent days, heterocycles and their derivatives have become strong reflection in medicinal research and pharmaceutical fields because of their practical pharmacological and biological activities.
Makkar, Reena, Sharma, Praveen Kumar
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Bazı α -lipoik asit türevi 1,3,4-tiyadiazol bileşiklerinin sentezi, karakterizasyonu ve antioksidan aktivitelerinin incelenmesi [PDF]
, 2021 Bu tez çalışmasında, kimyanın pek çok alanında olduğu gibi, özellikle endüstride, tıp ve eczacılıkta geniş kulanım alanlarına sahip olan 1,3,4-tiyadiazol bileşiklerinden, α-lipoik asit türevi tiyadiazol bileşikleri sentezi, karakterizasyonu ve ...
Mohammed Alı Abraheem, Ashweeqı
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Chemical and Pharmaceutical Bulletin, 1958 1) 1-(5-R-1, 3, 4-Thiadiazol-2-yl)-3-methyl-4-R'-2-pyrazolin-5-one (R'=H, iso-C3H7) (III) were synthesized starting with 2-hydrazino-5-R-1, 3, 4-thiadiazole (I : R=CH3, C2H5, n-C3H7, iso-C4H9, C6H5), and reacting them with ethyl acetoacetate or ethyl 3-acetyliso-valerate to form 5-R-1, 3, 4-thiadiazolylhydrazone (II).
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Modular Donor‐Acceptor Diradicaloids Based on an Electron Deficient N‐Heteroacene Acceptor
Small, Volume 22, Issue 20, 7 April 2026.This work presents a modular approach to donor‐acceptor‐donor (D‐A‐D) diradicaloids that show systematic evolution of their energy gaps, singlet‐triplet splittings, and diradical character (y). The correlation of (opto)electronic, spin, and magnetic properties with high‐fidelity theoretical investigations provides clear connections between the degree ...
Tanner L. Smith +9 more
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Synthesis and Preliminary Antibacterial Study of New 2-Mercapto-1, 3- Benzothiazole DerivativesWith Expected Biological Activity [PDF]
, 2013 Benzothiazoles are bicyclic ring system which have multiple applications. as antitumor , antiviral , antibacterial , anthelmintic and some of them showed glucose level.20 lowering effect. Accordingly, research is conducted to synthesize and evaluate some
Samer Abbas Ali
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Angewandte Chemie, Volume 138, Issue 14, 27 March 2026.A modular two‐step strategy provides tetraaza[n]helicenes (n = 7–15) as a homologous series with tunable photophysical and chiroptical properties. Extension beyond n = 11 induces pronounced through‐space π–π interactions, narrowing the energy gap and amplifying circularly polarized luminescence.
Takashi Otani +6 more
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Synthesis, characterization and cyclization reactions of some new bisthiosemicarbazones [PDF]
, 2009 The reaction of trans-1, 4-dichloro-2-butene 1 with selected phenols affords (E)-1, 4-bis(aryloxy)-2-butenes 2a-d which are converted into bis-thiosemicarbazones 3a-h via the reactions with thiosemicarbazide and 4-methyl thiosemicarbazide, respectively ...
Değirmencioğlu, İsmail +4 more
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Recent advances in the development of tissue transglutaminase (TG2) inhibitors [PDF]
, 2013 Tissue transglutaminase (TG2) is a Ca2+-dependent enzyme and probably the most ubiquitously expressed member of the mammalian transglutaminase family. TG2 plays a number of important roles in a variety of biological processes.
Badarau, Eduard +2 more
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Drug Design, Development and Therapy, 2018 Sobhi M Gomha,1 Mastoura M Edrees,2,3 Zeinab A Muhammad,2 Ahmed AM El-Reedy4 1Department of Chemistry, Faculty of Science, Cairo University, Giza, Egypt; 2Department of Organic Chemistry, National Organization for Drug Control and Research (NODCAR ...
Gomha SM +3 more
doaj
Synthesis, crystal structure, DFT and molecular docking studies of N-acetyl-2,4-[diaryl-3-azabicyclo[3.3.1]nonan-9-yl]-9-spiro-4'-acetyl-2'-(acetylamino)-4',9-dihydro-[1',3',4']-thiadiazoles: A potential SARS-nCoV-2 Mpro (COVID-19) inhibitor. [PDF]
J Mol Struct, 2022 Rajamanickam R +4 more
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