Results 71 to 80 of about 3,896 (275)
E-Journal of Chemistry, 2011 In the present study we report the synthesis and antibacterial activity of a new series 2-(1-methyl-4-nitro-1H-imidazol-5-ylsulfonyl)-1,3,4-thiadiazoles (6a-c).
Bahram Letafat +3 more
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BMC Cancer, 2017 Background Expression and activity of heparanase, an endoglycosidase that cleaves heparan sulfate (HS) side chains of proteoglycans, is associated with progression and poor prognosis of many cancers which makes it an attractive drug target in cancer ...
C. P. Baburajeev +9 more
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Synthesis and Biological evalution of some substituted 2-dibenzyl amino 1,3,4-oxadiazoles , thiadiazoles and 1,2,4-triazoles [PDF]
مجلة التربية والعلم, 2013 In this paper the synthesis of some substituted 2-dibenzyl 1,3,4-oxadiazole, thiadiazole and 1,2,4-triazoles derived from dibenzyl amine is reported scheme-1.
Khalid Daoud, Shaima Ismmaeel
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Design, synthesis and biological evaluation of novel thiadiazoline-thiazolone hybrids as kinase inhibitors. [PDF]
, 2017 Masters Degree. University of KwaZulu-Natal, Durban. 2017Cancer is a leading cause of death globally, and it was responsible for 8.8 million deaths in 2015. It is predicted that there will be 22 million new cancer cases by 2030 worldwide. Approximately,
Khathi, Samukelisiwe Pretty.
core
Anti-Candida and anti-quorum sensing activity of airborne microorganisms detected by a rapid method [PDF]
, 2022 Introduction: Introducing new antibiotics to the clinic is critical. Methods: We adapted a plate method described by Kawaguchi and coworkers in 20131 for detecting inhibitory airborne microorganisms.
Cruz, Andria Lopes +1 more
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Dual‐Phosphorus, Dual‐Nitrogen‐Embedded Corannulene: Synthesis, Structure, and Electronic Coupling
ChemistryEurope, Volume 4, Issue 5, May 2026.P2N2‐TBC, a corannulene‐based bowl structure incorporating two phosphorus and two nitrogen atoms, represents the first P2N2‐embedded heterobuckybowl. The cis and trans stereoisomers of this compound display distinct packing motifs, leading to markedly different electronic coupling patterns.
Marina Nagai +6 more
wiley +1 more source
3-(2-Fluorophenyl)-6-(phenoxymethyl)-1,2,4-triazolo[3,4-b][1,3,4]thiadiazole
Acta Crystallographica Section E, 2008 The crystal structure of the title compound, C16H11FN4OS, was synthesized in the course of our studies on 1,2,4-triazolo[3,4-b][1,3,4]thiadiazoles as inhibitors of p38 mitogen-activated protein kinase (MAPK). The three-dimensional data obtained were used
Stefan Laufer +2 more
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Synthesis of some substituted 1,3,4-oxadiazoles, 1,3,4-thiadiazoles and 1,2,4-triazoles from 2-(2,3-dimethylphenyl amino) benzoic acid [PDF]
مجلة التربية والعلم, 2009 In this paper the synthesis of some substituted 1,3,4-oxadiazoles, 1,3,4-thiadiazoles and 1,2,4-triazoles was achieved. 2-(2,3-dimethyl phenyl amino) benzoic acid was esterified to its ethyl ester by its reaction with absolute ethanol in presence of ...
Khalid Daoud +2 more
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ChemistryOpen, Volume 15, Issue 5, May 2026.In this present study, an enzyme‐based amperometric nanobiosensor was designed and fabricated through the immobilization of tyrosinase onto a selenium‐bearing conducting polymer (poly[BDT‐alt‐(TP;BSe)]), in combination with NH2‐functionalized graphene quantum dots incorporating benzoselenadiazole, thienopyrroledione, and benzodithiophene moieties.
Raghad Alhardan +8 more
wiley +1 more source
Synthesis and Preliminary Antimicrobial Study of 2-Amino-5-Mercapto-1,3,4-Thiadiazole Derivatives
Iraqi Journal of Pharmaceutical Sciences, 2017 Nitrogen heterocycles are of a special interest because they constitute an important class of natural and non natural products, many of which exhibit useful biological activities.Among these nitrogen heterocycles are 1, 3, 4-thiadiazole containing ...
Husam A. Ameen, Ahlam J. Qasir
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