Results 81 to 90 of about 2,685 (205)

MOLECULAR DOCKING STUDIES ON THIADIAZOLE DERIVATIVES AS PROTEIN KINASE INHIBITORS [PDF]

, 2018
Objective: In the present study, a novel series of 1, 3, 4-thiadiazole derivatives were docked against the mycobacterium tuberculosis protein kinase G.
Geetha, G., Sivakumar, D.
core   +1 more source

Synthesis and Characterization New 1, 2, 4-Triazole Derivative and Its Complexes with Some Transition Metal Ions [PDF]

An innovative class of ligand compounds using The ions of transition metals (Cr(III), Fe(III), and Ni(II)).The ligand N,N'-(4H-1,2,4-triazole-3,5-diyl)bis(4-methoxybenzamide) was produced by reacting 2,5-di amino-1,2,4-triazole with two moles of methyl 4-
Natheil, Amal Hussein
core   +2 more sources

Exploring Novel Nitrofuryl‐1,3,4‐Thiadiazole‐Based Derivatives: Design, Synthesis, and Evaluation of In Vitro Leishmanicidal and Trypanocidal Activity

Archiv der Pharmazie, Volume 359, Issue 3, March 2026.
In a series of substituted 1‐[5‐(5‐nitrofuran‐2‐yl)‐1,3,4‐thiadiazol‐2‐yl]piperidine‐4‐carboxamides evaluated for in vitro antileishmanial and antitrypanosomal activity, compound 18 emerged as the most promising derivative, showing submicromolar anti‐parasitic effects targeting diverse Leishmania and Trypanosoma species and acceptable selectivity ...
Alireza Mousavi, Martina Slapničková, Maryam Norouzbahari, Sarah D'Alessandro, Parham Foroumadi, Fariba Peytam, Federica Perego, Eva Doleželová, Zahra Emamgholipour, Maliheh Barazandeh Tehrani, Seyed Esmaeil Sadat‐Ebrahimi, Elahe Hosseinzadeh, Elmira Meghrazi Ahadi, Loghman Firoozpour, Hamidreza Bijanzadeh, Nicoletta Basilico, Alena Zíková, Alireza Foroumadi   +17 more
wiley   +1 more source

Synthesis, characterization and cyclization reactions of some new bisthiosemicarbazones [PDF]

, 2009
The reaction of trans-1, 4-dichloro-2-butene 1 with selected phenols affords (E)-1, 4-bis(aryloxy)-2-butenes 2a-d which are converted into bis-thiosemicarbazones 3a-h via the reactions with thiosemicarbazide and 4-methyl thiosemicarbazide, respectively ...
Değirmencioğlu, İsmail, Er, Mustafa, Karaoğlu, Şengül Alpay, Sancak, Kemal, Ünver, Yasemin   +4 more
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Nitrogen‐Doped Graphene Aerogels for Supercapacitors: Advances in Synthesis and Electrochemical Performance

Battery Energy, Volume 5, Issue 2, March 2026.
This review explores nitrogen‐doped graphene aerogel materials used in supercapacitors, analyzing synthesis techniques, performance measures, and recent advancements. It highlights material challenges and limitations while suggesting directions for future research.
Khaled Abdou Ahmed Abdou Elsehsah, Zulkarnain Ahmad Noorden, Norhafezaidi Mat Saman, Noor Azlinda Ahmad, Mohd Faizal Hasan, Sharin Ab Ghani, Ayaz Ahmed   +6 more
wiley   +1 more source

5-(Thiophen-2-yl)-1,3,4-thiadiazole derivatives: synthesis, molecular docking and in vitro cytotoxicity evaluation as potential anticancer agents

Drug Design, Development and Therapy, 2018
Sobhi M Gomha,1 Mastoura M Edrees,2,3 Zeinab A Muhammad,2 Ahmed AM El-Reedy4 1Department of Chemistry, Faculty of Science, Cairo University, Giza, Egypt; 2Department of Organic Chemistry, National Organization for Drug Control and Research (NODCAR ...
Gomha SM, Edrees MM, Muhammad ZA, El-Reedy AA   +3 more
doaj  

Synthesis and Preliminary Antibacterial Study of New 2-Mercapto-1, 3- Benzothiazole DerivativesWith Expected Biological Activity [PDF]

, 2013
Benzothiazoles are bicyclic ring system which have multiple applications. as antitumor , antiviral , antibacterial , anthelmintic and some of them showed glucose level.20 lowering effect. Accordingly, research is conducted to synthesize and evaluate some
Samer Abbas Ali
core   +2 more sources

Synthesis of Related Compounds of Thiosemi-carbazide. IV. 1-(1, 3, 4-Thiadiazol-2-yl)-2-pyrazolin-5-one and Tetrazolo [4, 5-a]-1, 3, 4-thiadiazole Derivatives.

Chemical and Pharmaceutical Bulletin, 1958
1) 1-(5-R-1, 3, 4-Thiadiazol-2-yl)-3-methyl-4-R'-2-pyrazolin-5-one (R'=H, iso-C3H7) (III) were synthesized starting with 2-hydrazino-5-R-1, 3, 4-thiadiazole (I : R=CH3, C2H5, n-C3H7, iso-C4H9, C6H5), and reacting them with ethyl acetoacetate or ethyl 3-acetyliso-valerate to form 5-R-1, 3, 4-thiadiazolylhydrazone (II).
openaire   +3 more sources

Structural design and property regulation of organic polymers for photocatalytic synthesis of H2O2

InfoScience, Volume 3, Issue 1, March 2026.
Photocatalytic synthesis of H2O2 offers a sustainable approach. Photocatalytic efficiency depends critically on interfacial electron transfer kinetics and spatial charge separation. Herein, we systematically analyze key factors governing photogenerated carrier dynamics and propose engineered strategies to optimize performance, thereby providing design ...
Mingyang Xu, Rongchen Shen, Yingyin Mo, Guijie Liang, Shijie Li, Peng Zhang, Xiaobo Chen, Youji Li, Xin Li   +8 more
wiley   +1 more source

Bazı α -lipoik asit türevi 1,3,4-tiyadiazol bileşiklerinin sentezi, karakterizasyonu ve antioksidan aktivitelerinin incelenmesi [PDF]

, 2021
Bu tez çalışmasında, kimyanın pek çok alanında olduğu gibi, özellikle endüstride, tıp ve eczacılıkta geniş kulanım alanlarına sahip olan 1,3,4-tiyadiazol bileşiklerinden, α-lipoik asit türevi tiyadiazol bileşikleri sentezi, karakterizasyonu ve ...
Mohammed Alı Abraheem, Ashweeqı
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