Results 91 to 100 of about 23,173 (263)

Synthesis and In Vitro Anticancer Activity of Pyrrolidone Derivatives Bearing 3,4,5-Trimethoxyphenyl Moiety as a Promising Anticancer Scaffold

Applied Sciences
A series of 5-oxo-1-(3,4,5-trimethoxyphenyl)pyrrolidine-3-carboxylic acid derivatives–hydrazones, N-ethylhydrazones, pyrrole, pyrazole, oxadiazole, and triazole were synthesized and evaluated for their anticancer activity using human A549 pulmonary ...
Povilas Kavaliauskas, Birutė Sapijanskaitė-Banevič, Birutė Grybaitė, Eglė Mickevičiūtė, Kazimieras Anusevičius, Andrew Garcia, Ethan Naing, Rūta Petraitienė, Vidmantas Petraitis, Ramunė Grigalevičiūtė, Vytautas Mickevičius   +10 more
doaj   +1 more source

Disease control in oilseed rape: Current insights and perspectives for next‐generation integrated pest management

Pest Management Science, EarlyView.
Winter oilseed rape in Europe suffers frequent pathogen losses. This review outlines key integrated pest management (IPM) strategies, rotation, residue and tillage management, optimized sowing, resistance, and targeted fungicides supported by forecasting.
Jon S West, Małgorzata Jędryczka, Nazanin Zamani‐Noor   +2 more
wiley   +1 more source

Mutación r30q en cyp51a de neocosmospora solani asociada a resistencia a azoles [PDF]

, 2021
Neocosmospora and Fusarium are the etiological agents of human fusariosis such as onychomycosis, fungal keratitis and disseminated infections, and the most widely reported species are Neocosmospora keratoplastica, Neocosmospora falciformis and Fusarium ...
Lizcano Salas, Andrés Felipe
core  

Corrosion Protection of Copper Using Azoles Applied on Its Surface at High Temperature Under Vacuum

International Journal of Electrochemical Science, 2011
Application of seven different azoles namely; 1H-Pyrazole-3,5-diamine (azole 1), 1-Benzoyl benzotriazole (azole 2), 1-P-Chloro-Benzoyl benzotriazole (azole3), 1-P-Methoxy-Benzoyl benzotriazole (azole 4), 4-Phenyl-1H-pyrazole-3,5-diamine (azole5), N ...
F. M. Al Kharafi, N.A. Al-Awadi, I.M. Ghayad, R.M. Abdullah, M.R. Ibrahim   +4 more
doaj   +1 more source

DFT investigations on arylsulphonyl pyrazole derivatives as potential ligands of selected kinases

Open Chemistry, 2020
Using the density functional theory (DFT) formalism, we have investigated the properties of some arylsulphonyl indazole derivatives that we studied previously for their biological activity and susceptibility to interactions of azoles. This study includes
Czaja Kornelia, Kujawski Jacek, Kujawski Radosław, Bernard Marek K.   +3 more
doaj   +1 more source

The continuing significance of chiral agrochemicals

Pest Management Science, Volume 81, Issue 4, Page 1697-1716, April 2025.
In the time frame 2018–2023, around 43% of the 35 chiral agrochemicals introduced to the market (herbicides, fungicides, insecticides, acaricides, and nematicides) contain one or more stereogenic centers in the molecule, and almost 69% of them have been marketed as racemic mixtures of enantiomers or stereoisomers.
Peter Jeschke
wiley   +1 more source

Substituent effects on the N-15 MMR parameters of azoles [PDF]

, 1997
Substituent eþ ects on the 15N NMR compounds in several solvents were Parameters of Azoles recorded again and 31 compounds were ROSA CLARAMUNT, DIONI-MARIŠ A SIA SANZ, andCONCEPCIOŠ NLOŠ PEZ JOSE ANTONIOŠ JIMEŠ NEZ studied for the first time;
Elguero, José, Sanz, Dionisia, Jimeno, M. Luisa, Jiménez, José Antonio, Fruchier, Alain, Claramunt, Rosa M., López, Concepción   +6 more
core  

Virulence factors of Candida spp and molecular mechanisms of resistance to azoles expressed by Candida tropicalis [PDF]

Introducción: Debido al panorama epidemiológico de la candidiasis producida por Candida tropicalis y la marcada resistencia generada hacia los azoles, se hace necesario profundizar en el conocimiento de la virulencia y mecanismos de resistencia a ...
Cárdenas Parra, Leidy Yurany, Rojas Rodríguez, Ana Elisa, Zapata Serna, Yuliana, Pérez Cárdenas, Jorge Enrique   +3 more
core   +2 more sources

Uptake of azoles by lamb's lettuce (Valerianella locusta L.) grown in hydroponic conditions [PDF]

, 2016
An uptake and translocation study of azole compounds was performed in lamb's lettuce (Valerianella locusta L.) grown in nutrient solution fortified with different azoles.
Escorial, Concepción, Tadeo Lluch, José Luis, Molero Vega, M. Encarnación, García Valcárcel, Ana Isabel, Loureiro, Íñigo   +4 more
core   +1 more source

Real‐world outcomes of triplet therapy with gilteritinib, azacitidine and venetoclax in FMS‐like tyrosine kinase 3 (FLT3)‐mutated relapsed/refractory acute myeloid leukaemia: A UK single‐centre experience

British Journal of Haematology, EarlyView.
In FMS‐like tyrosine kinase 3 (FLT3)‐mutated relapsed/refractory acute myeloid leukaemia, gilteritinib, azacitidine and venetoclax is an effective salvage option with an ORR of 100% (mCRc [MLFS + CRc] 93%). Sixty‐two per cent of patients treated with intention‐to‐transplant proceeded to allogeneic haematopoietic stem cell transplant, of whom 50% remain
Wei Yee Chan, Hannah Al‐Yousuf, Ho Pui Jeff Lam, Sarah Leong, Jiexin Zheng, Richard Burt, Andrew J. Wilson, Ke Xu, Kate Stringaris, Samah Alimam, Kavita Raj, Rajeev Gupta, Panagiotis Kottaridis, Anish Tailor, Rebecca Burgoyne, Marc R. Mansour, Asim Khwaja, Rob Sellar, Elspeth M. Payne, Jenny O'Nions   +19 more
wiley   +1 more source