Results 81 to 90 of about 23,046 (254)
3D-QSAR and pharmacophore model study on aryl diphenolic azoles as estrogen receptor-b ligands
, 2013 3D-QSAR and pharmacophore model study on aryl diphenolic azoles as estrogen receptor-b ...
Jun-Zhi Wang +4 more
core
Direct, Regioselective N‑Alkylation of 1,3-Azoles
, 2016 Regioselective N-alkylation of 1,3-azoles is a valuable transformation. Organomagnesium reagents were discovered to be competent bases to affect regioselective alkylation of various 1,3-azoles. Counterintuitively, substitution selectively occurred at the
Alessandro A. Boezio (1447501) +2 more
core +1 more source
A General Copper-Catalyzed Coupling of Azoles with Vinyl Bromides
, 2016 A copper-catalyzed methodology for the coupling of vinyl bromides with azoles has been developed. This protocol uses a combination of 10 mol % of copper iodide and 20 mol % of ethylenediamine as catalyst.
Qian Liao (1489453) +3 more
core +1 more source
Palladium-Catalyzed Direct Oxidative Alkenylation of Azoles
, 2016 The direct heteroaromatic sp2 C−H alkenylation of 2-substituted azole compounds with alkenes proceeds in the presence of Pd(OAc)2 and AgOAc as catalyst and oxidant, respectively, to afford the corresponding 5-alkenylated azoles in good ...
Mitsuru Miyasaka (2233909) +3 more
core +1 more source
Frontiers in Microbiology, 2018 Objectives: Invasive mold infections associated with Aspergillus species are a significant cause of mortality in immunocompromised patients. The most frequently occurring aetiological pathogens are members of the Aspergillus section Fumigati followed by ...
Tamara Zoran +53 more
doaj +1 more source
DFT investigations on arylsulphonyl pyrazole derivatives as potential ligands of selected kinases
Open Chemistry, 2020 Using the density functional theory (DFT) formalism, we have investigated the properties of some arylsulphonyl indazole derivatives that we studied previously for their biological activity and susceptibility to interactions of azoles. This study includes
Czaja Kornelia +3 more
doaj +1 more source
Pest Management Science, EarlyView.For three collections of Irish Pyrenopeziza brassicae populations fungicide sensitivity status to methyl benzimidazole carbamate (MBC), quinone outside inhibitor (QoI) and succinate dehydrogenase inhibitor (SDHI) fungicides was determined using sensitivity screening in vitro. Molecular mechanisms of insensitivity have been identified for MBC and QoI in
Diana E Bucur +3 more
wiley +1 more source
AntibioticsBackground/Objectives: Malassezia pachydermatis is a lipophilic yeast frequently associated with otitis externa and dermatological disorders in companion animals. This study aimed to evaluate the antifungal susceptibility of M.
Marianna Domán +5 more
doaj +1 more source
Memorias do Instituto Oswaldo Cruz, 2012 Ketoconazole is a clinically safe antifungal agent that also inhibits the growth of Leishmania spp. A study was undertaken to determine whether Leishmania parasites are prone to becoming resistant to ketoconazole by upregulating C14-demethylase after ...
Valter Viana Andrade-Neto +5 more
doaj +1 more source
The continuing significance of chiral agrochemicals
Pest Management Science, Volume 81, Issue 4, Page 1697-1716, April 2025.In the time frame 2018–2023, around 43% of the 35 chiral agrochemicals introduced to the market (herbicides, fungicides, insecticides, acaricides, and nematicides) contain one or more stereogenic centers in the molecule, and almost 69% of them have been marketed as racemic mixtures of enantiomers or stereoisomers.
Peter Jeschke
wiley +1 more source