Results 51 to 60 of about 24,787 (257)

Serotonin 5-HT4 Agonist Activity of a Series of Meso-Azanoradamantane Benzamides [PDF]

, 1997
A series of meso-amino(methyl)azanoradamantane benzamides has been prepared and evaluated for 5-HT4agonism activity in the rat tunica muscularis mucosae (TMM) assay.
Becker, Daniel, Gullikson, Gary, Nosal, Roger, Villamil, Clara I.   +3 more
core   +1 more source

4-Iodo-N-(phenylsulfonyl)benzamide hemihydrate

IUCrData, 2017
In the title hemihydrate, 2C13H10INO3S·H2O, there are two organic molecules (A and B) and one water molecule in the asymmetric unit. The benzene rings are inclined to one another by 77.98 (1)° in A and 79.81 (9)° in B. The A and B molecules are connected
P. A. Suchetan, A. G. Sudha, E. Suresha, N. K. Lokanath, S. Naveen, Ismail Warad   +5 more
doaj   +1 more source

4-Bromo-N-(diisopropoxyphosphoryl)benzamide [PDF]

Acta Crystallographica Section E Structure Reports Online, 2009
In the title compound, C(13)H(19)BrNO(4)P, the crystal structure is stabilized by inter-molecular N-H⋯O hydrogen bonds between the phosphoryl O atom and the amide N atom which link the mol-ecules into centrosymmetric dimers. These dimers are further packed into stacks along the c axis by inter-molecular C-H⋯O and C-H⋯π inter-actions.
Strasser C.E., Sheng X., Safin D.A., Raubenheimer H.G., Luckay R.C.   +4 more
openaire   +6 more sources

Towards a Sequential One-Pot Preparation of 1,2,3-Benzotriazin-4(3H)-ones Employing a Key Cp*Co(III)-catalyzed C-H Amidation Step [PDF]

, 2018
1,2,3‐benzotriazin‐4(3H)‐one derivatives have been recognised for their potential application as pesticides and pharmaceuticals and new methodologies for their preparation, starting from readily accessible reagents would therefore be an attractive ...
Anastas, Bariwalab, Barsu, Bunno, Campbell, Chirila, Chirila, Davies, Evano, Gensch, Hayashi, Hili, Huang, Hwang, Ibrahim, Jiao, Kawade, Khalid, Li, Liang, Lu, Mei, Miura, Miura, Moselage, Park, Park, Patel, Pototschnig, Prakash, Qin, Qu, Ruiz-Castillo, Shi, Shin, Simmons, Sun, Sun, Sun, Tan, Thorat, Wan, Wang, Wang, Wang, Wang, Wang, Wang, Wei, Wencel-Delord, Whiteoak, Yedage, Yi, Yoshino, Yoshino, Yoshino, Yu, Zhu   +57 more
core   +1 more source

A two-step approach to achieve secondary amide transamidation enabled by nickel catalysis. [PDF]

, 2016
A long-standing challenge in synthetic chemistry is the development of the transamidation reaction. This process, which involves the conversion of one amide to another, is typically plagued by unfavourable kinetic and thermodynamic factors. Although some
Anthony, Sarah M, Baker, Emma L, Garg, Neil K, Yamano, Michael M, Zhou, Yujing   +4 more
core   +2 more sources

Synthesis, Spectroscopic Properties and Antipathogenic Activity of New Thiourea Derivatives

Molecules, 2011
A number of acylthioureas, 2-((4-methylphenoxy)methyl)-N-(aryl-carbamothioyl)benzamides (aryl = 3,5-dichlorophenyl, 2,3-dichlorophenyl, 3,4-dichloro-phenyl, 2,4,5-trichlorophenyl, 3,4,5-trichlorophenyl, 2-bromophenyl, 2,4-dibromophenyl, 2,5-dibromophenyl,
Carmen Limban, Luminita Marutescu, Mariana Carmen Chifiriuc   +2 more
doaj   +1 more source

The PIFA-initiated oxidative cyclization of 2-(3-butenyl)quinazolin-4(3H)-ones – an efficient approach to 1-(hydroxymethyl)-2,3-dihydropyrrolo[1,2-a]quinazolin-5(1H)-ones

Beilstein Journal of Organic Chemistry, 2021
A regioselective method for the synthesis of 1-(hydroxymethyl)-2,3-dihydropyrrolo[1,2-a]quinazolin-5(1H)-ones – close structural analogs of naturally occurring vasicinone alkaloids – is described.
Alla I. Vaskevych, Nataliia O. Savinchuk, Ruslan I. Vaskevych, Eduard B. Rusanov, Oleksandr O. Grygorenko, Mykhailo V. Vovk   +5 more
doaj   +1 more source

N-(Pyrrolidin-1-ylcarbothioyl)benzamide [PDF]

Acta Crystallographica Section E Structure Reports Online, 2011
In the title compound, C(12)H(14)N(2)OS, the pyrrolidine ring adopts an envelope conformation with the C atom at the 3-position as the flap and makes a dihedral angle of 65.80 (9)° with the benzene ring. In the crystal, N-H⋯O hydrogen bonds join c-glide related mol-ecules into chains extended along [001] that are further connected into (100) layers via
Al-Abbasi, Aisha A., Mohamed Tahir, Mohamed Ibrahim, Kassim, Mohammad   +2 more
openaire   +3 more sources

N-(INDAZOLYL)BENZAMIDO DERIVATIVES AS CDK1 INHIBITORS: DESIGN, SYNTHESIS, BIOLOGICAL ACTIVITY, AND MOLECULAR DOCKING STUDIES [PDF]

, 2009
A series of N-1H-indazole-1-carboxamides have been synthesized and their effects on both CDK1/cyclin B and K-562 (human chronic myelogenus leukemia) cell line were evaluated.
Arris, Candurri, Candurri, Carmicael, Daidone, Davies, Davies, de Azevedo, Fabbro, Furet, Gray, Jeffrey, Knockaert, Korbonits, Manfredini, McGrath, Raffa, Raffa, Schulze-Gahmen, Smith, Toogood, Valgeirsson   +21 more
core   +1 more source

N-(4-Cyanobenzyl)benzamide

Acta Crystallographica Section E Structure Reports Online, 2008
The title compound, C(15)H(12)N(2)O, is a derivative of 4-(amino-meth-yl)benzonitrile, an important pestcide inter-mediate. In the crystal structure, mol-ecules are linked via inter-molecular N-H⋯O hydrogen bonds, forming infinite chains.
Hong-Jun Zhu, Wei Chen, Hai-Jun Ma, Li-Qin Guo, Yi-Li Tong   +4 more
openaire   +3 more sources