Results 131 to 140 of about 104,722 (190)

Exploring Carbon Nanomaterial Diversity for Nucleation of Protein Crystals [PDF]

, 2015
Chain B, Chayen, N, Govada, Hu S, Kassen, Khurshid, Leese H S, Menzel, Saridakis, Shaffer   +9 more
core   +1 more source

Development of cell-active BRD4-D1 selective inhibitors to decode the role of BET proteins in LPS-mediated liver inflammation. [PDF]

Eur J Med Chem
Scholtz CR, Doskey LC, Kandanur SGS, Vail NR, Roderick ER, Peterson EJ, Hoell ZJ, Shi K, Aihara H, Kostallari E, Shah VH, Malhi H, Pomerantz WCK.   +12 more
europepmc   +1 more source

A "Goldilocks Zone" for Recruiting BET Proteins with Bromodomain-1-Selective Ligands. [PDF]

ACS Chem Biol
Mohammed A, Churion K, Danda A, Philips SJ, Ansari AZ.   +4 more
europepmc   +1 more source

PRC2 loss of function confers a targetable vulnerability to BET proteins in T-ALL.

Blood, 2021
Andrieu GP, Kohn M, Simonin M, Smith CL, Cieslak A, Dourthe MÉ, Charbonnier G, Graux C, Huguet F, Lhéritier V, Dombret H, Spicuglia S, Rousselot P, Boissel N, Asnafi V.   +14 more
europepmc   +1 more source

Selective targeting of BD1 and BD2 of the BET proteins in cancer and immunoinflammation. [PDF]

Science, 2020
Gilan O, Rioja I, Knezevic K, Bell MJ, Yeung MM, Harker NR, Lam EYN, Chung CW, Bamborough P, Petretich M, Urh M, Atkinson SJ, Bassil AK, Roberts EJ, Vassiliadis D, Burr ML, Preston AGS, Wellaway C, Werner T, Gray JR, Michon AM, Gobbetti T, Kumar V, Soden PE, Haynes A, Vappiani J, Tough DF, Taylor S, Dawson SJ, Bantscheff M, Lindon M, Drewes G, Demont EH, Daniels DL, Grandi P, Prinjha RK, Dawson MA.   +36 more
europepmc   +1 more source

Inhibition of BET proteins modulates amyloid-beta accumulation and cognitive performance in middle-aged mice prenatally exposed to maternal immune activation. [PDF]

Front Mol Neurosci
Matuszewska M, Wilkaniec A, Gąssowska-Dobrowolska M, Cieślik M, Olech-Kochańczyk G, Pałasz E, Gawinek E, Strawski M, Czapski GA.   +8 more
europepmc   +1 more source

BET proteins: Investigating BRDT as a potential target for male contraception. [PDF]

Bioorg Med Chem Lett, 2020
Wisniewski A, Georg GI.
europepmc   +1 more source

Targeted inhibition of BET proteins in HPV16-positive head and neck squamous cell carcinoma reveals heterogeneous transcriptional responses. [PDF]

Front Oncol
Rao A, Stosic MS, Mohanty C, Suresh D, Wang AR, Lee DL, Nickel KP, Chandrashekar DS, Kimple RJ, Lambert PF, Kendziorski C, Rounge TB, Iyer G.   +12 more
europepmc   +1 more source

Correction: Comparative structure-function analysis of bromodomain and extraterminal motif (BET) proteins in a gene-complementation system. [PDF]

J Biol Chem, 2020
Werner MT, Wang H, Hamagami N, Hsu SC, Yano JA, Stonestrom AJ, Behera V, Zhong Y, Mackay JP, Blobel GA.   +9 more
europepmc   +1 more source

Brd/BET Proteins Influence the Genome-Wide Localization of the Kaposi's Sarcoma-Associated Herpesvirus and Murine Gammaherpesvirus Major Latency Proteins. [PDF]

Front Microbiol, 2020
Lotke R, Schneeweiß U, Pietrek M, Günther T, Grundhoff A, Weidner-Glunde M, Schulz TF.   +6 more
europepmc   +1 more source