Results 141 to 150 of about 5,584 (214)

The thiazolidinedione drug troglitazone inhibits Gq signaling through direct binding to the Gq alpha subunit through inhibition of GDP release. [PDF]

Mol Pharmacol
Issa NT, Shen T, Vizurraga A, Pronin A, Henry T, Wang Q, Kwarcinski FE, Schürer S, Badiavas E, Tall GG, Slepak VZ.   +10 more
europepmc   +1 more source

Total Synthesis of Marformycins A and D. [PDF]

Org Lett
Anwar AF, Elbatrawi YM, Degen D, Ebright RH, Del Valle JR.   +4 more
europepmc   +1 more source

Biosynthesis of the Fungal Cyclic Lipodepsipeptide Pleosporacin, a New Selective Inhibitor of the Phytopathogen Botrytis cinerea. [PDF]

Chembiochem
Wieder C, Wiechert R, Yemelin A, Sandjo LP, Thines E, Opatz T, Schüffler A.   +6 more
europepmc   +1 more source

End-to-End Backbone Cyclization Enhances Passive Permeability of bRo5 Oligomeric Depsipeptides with Nonlinear Size Dependence. [PDF]

ACS Med Chem Lett
Thorpe MP, Hopkins CR, Johnston JN.
europepmc   +1 more source

Current issues in heartworm chemotherapy. [PDF]

Parasit Vectors
Geary TG.
europepmc   +1 more source

Beauvericin Induces Mitochondrial Apoptosis and Attenuates EMT-Associated Phenotypes and Angiogenic Signaling in Colorectal Cancer Cells <i>In Vitro</i>. [PDF]

J Microbiol Biotechnol
Kwon M, Jung HJ.
europepmc   +1 more source

Cyclic peptide inhibitors function as molecular glues to stabilize Gq/11 heterotrimers. [PDF]

Proc Natl Acad Sci U S A
Mühle J, Alenfelder J, Rodrigues MJ, Jürgenliemke L, Guixà-González R, Grätz L, Andres F, Bacchin A, Hennig M, Schihada H, Crüsemann M, König GM, Schertler G, Kostenis E, Deupi X.   +14 more
europepmc   +1 more source

Amino acid analogues provide multiple plausible pathways to prebiotic peptides. [PDF]

J R Soc Interface
Zhang L, Ying J.
europepmc   +1 more source

Depsipeptide cyclisation: Lactonization vs. Lactamisation

Proceedings of the 35th European Peptide Symposium, 2018
Sacha Stadelmann, Stéphane Mayor, Roger Marti, Marc Mathieu   +3 more
openaire   +1 more source

Environmental metabolomics characterization of modern stromatolites and annotation of ibhayipeptolides. [PDF]

PLoS One
Neuhaus GF, Aron AT, Isemonger EW, Petras D, Waterworth SC, Madonsela LS, Gentry EC, Siwe Noundou X, Kalinski JJ, Polyzois A, Habiyaremye JC, Redick MA, Kwan JC, Dorrington RA, Dorrestein PC, McPhail KL.   +15 more
europepmc   +1 more source