Results 1 to 10 of about 7,968 (196)
Mechanistic DFT Study of 1,3-Dipolar Cycloadditions of Azides with Guanidine [PDF]
Molecules, 2023 Density functional calculations SMD(chloroform)//B3LYP/6-311+G(2d,p) were employed in the computational study of 1,3-dipolar cycloadditions of azides with guanidine.
Ivana Antol +2 more
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Self-Assembled Lipoplexes of Short Interfering RNA (siRNA) Using Spermine-Based Fatty Acid Amide Guanidines: Effect on Gene Silencing Efficiency [PDF]
Pharmaceutics, 2011 Four guanidine derivatives of N4,N9-diacylated spermine have been designed, synthesized, and characterized. These guanidine-containing cationic lipids bound siRNA and formed nanoparticles. Two cationic lipids with C18 unsaturated chains, N1,N12-diamidino-
Abdelkader A. Metwally +1 more
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Efficient Cleavage of pUC19 DNA by Tetraaminonaphthols [PDF]
ChemistryOpenIn an attempt to create models of phosphodiesterases, we previously investigated bis(guanidinium) naphthols. Such metal‐free anion receptors cleaved aryl phosphates and also plasmid DNA.
Catharina Kost +3 more
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Advanced glycation end products mediate biomineralization disorder in diabetic bone disease [PDF]
Cell Reports MedicineSummary: Patients with diabetes often experience fragile fractures despite normal or higher bone mineral density (BMD), a phenomenon termed the diabetic bone paradox (DBP).
Qianmin Gao +24 more
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Development of New Leishmanicidal Compounds via Bioconjugation of Antimicrobial Peptides and Antileishmanial Guanidines [PDF]
ACS Omega, 2023 Natalia C. S. Costa +8 more
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Synthesis of (+)-(R)-Tiruchanduramine
Molecules, 2022 The absolute stereochemistry of the marine alkaloid (+)-(R)-tiruchanduramine was established via a convergent total synthesis in six steps and 15.5% overall yield from Fmoc-D-Dab(Boc)-OH.
Zahraa S. Al-Taie +9 more
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Pharmaceuticals, 2023 This study examines the properties of novel guanidines, designed and synthesized as histamine H3R antagonists/inverse agonists with additional pharmacological targets.
Marek Staszewski +12 more
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Investigation of Disinfectant\u27s Effectiveness as to Contaminating Microflora in Sugar Production [PDF]
, 2018 The article presents the results of the studies of the effectiveness of disinfection means, based on chlorinated guanidines, tetradic ammonium salts, dichlorisocyanuric acid, peracetic acid and hydrogen peroxide as to the contaminating microflora of ...
Husiatynska, N. (Nataliia) +1 more
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Journal of Enzyme Inhibition and Medicinal Chemistry, 2023 A small library of substituted cyclic guanidine incorporated benzothiazole-6-sulphonamides was synthesized. All obtained compounds were investigated for their inhibitory activity against the key brain-associated human carbonic anhydrase isoform hCA VII ...
Morteza Abdoli +2 more
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Guanidinates as Alternative Ligands for Organometallic Complexes
Molecules, 2022 For decades, ligands such as phosphanes or cyclopentadienyl ring derivatives have dominated Coordination and Organometallic Chemistry. At the same time, alternative compounds have emerged that could compete either for a more practical and accessible ...
Fernando Carrillo-Hermosilla +3 more
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