Results 41 to 50 of about 562 (194)

Reactions with hydrazonoyl halides 65: Synthesis of some new 1,3,4-thiadiazoles and triazolino[4,3-a]pyrimidines containing pyrazole moiety [PDF]

, 2011
2,3-Dihydro-1,3,4-thiadiazoles, and triazolino[4,3-a]pyrimidines containing pyrazole moieties were prepared from the reaction of alkyl 2-[1-(4-cyano-1,5-diphenyl-1H-pyrazol-3-yl)ethylidene]hydrazinecarbodithioate and pyrimidine-2-thione derivatives with ...
Abdelhamid, Abdou Osman, Fahmi, Abdelgawad Ali, Halim, Karema Noury Mahmoud   +2 more
core   +1 more source

Synthesis, characterization and docking study of novel pyrimidine derivatives as anticancer agents [PDF]

, 2020
New compounds 5 and 9 using DNA bases e.g. Adenine 1 and Guanine 6 derivatives have been synthesized. The use of simple methods to synthesize compounds 5 and 9 were done using pyrimidine as an alternative DNA base ring.
El-Saidi, Manal Mohamed Talaat, El-Sayed, Ahmed Ali, Gad, Wafaa Ahmed, Mohamed, Nadia Ragab, Pedersen, Erik Bjerregaard, Tantawy, Mohamed Abdelhamid   +5 more
core   +1 more source

Synthesis, docking and evaluation of novel fused pyrimidine compounds as possible lead compounds with antibacterial and antitumor activities [PDF]

, 2023
Reaction of a series of hydrazonoyl chlorides with substituted aminopyrimidines afforded good selectivity in most cases leading either to formation of new imidazo[1,2-a]pyrimidine derivatives, or regioisomeric hydrazonamide adducts.
Abu-Teim, Omar S., Al-Reefi, Mariam R, Almasri, Ihab M., Alzaharna, Mazen M., Awadallah, Adel M., Azarah, Jannat N., Beadham, Ian, El-Hallaq, Amany F., Elmanama, Abdelraouf A., Gardiner, John M., Morjan, Rami Y., Raftery, James   +11 more
core   +1 more source

Synthesis and Antimicrobial Activity of Some New Thiadiazoles, Thioamides, 5-Arylazothiazoles and Pyrimido[4,5-d][1,2,4]triazolo[4,3-a]pyrimidines

Molecules, 2016
A novel series of 1,3,4-thiadiazoles, 5-arylazothiazoles and hexahydropyrimido-[4,5-d][1,2,4]triazolo[4,3-a]pyrimidines were synthesized via reaction of hydrazonoyl halides with each of alkyl carbothioates, carbothioamides and 7-thioxo-5,6,7,8 ...
Abdou O. Abdelhamid, Ibrahim E. El Sayed, Mohamed Z. Hussein, Mangoud M. Mangoud   +3 more
doaj   +1 more source

Synthesis and Cytotoxicity Evaluation of Some Novel Thiazoles, Thiadiazoles, and Pyrido[2,3-d][1,2,4]triazolo[4,3-a]pyrimidin-5(1H)-ones Incorporating Triazole Moiety

Molecules, 2015
Reactions of hydrazonoyl halides and each of methyl 2-(1-(5-methyl-1-phenyl-1H-1,2,3-triazol-4-yl)ethylidene)hydrazine-1-carbodithioate and 2-(1-(5-methyl-1-phenyl-1H-1,2,3-triazol-4-yl)ethylidene)hydrazine-1-carbothioamide afforded 2-(1-(5-methyl-1 ...
Sobhi M. Gomha, Sayed A. Ahmed, Abdou O. Abdelhamid   +2 more
doaj   +1 more source

Ultrasound-assisted green synthesis and antimicrobial assessment of 1,3-thiazoles and 1,3,4-thiadiazines

Green Chemistry Letters and Reviews, 2021
In this article, we applied ultrasonic irradiation as an ecofriendly, green, efficient approach for the synthesis of a new 1,3-thiazoles and 1,3,4-thiadiazines under solvent-free conditions.
Sara N. Shabaan, Basma Saad Baaiu, Anhar Abdel-Aziem, Mohamed S. Abdel-Aziz   +3 more
doaj   +1 more source

Reaction of nitrilimines and nitrile oxides with hydrazines, hydrazones and oximes [PDF]

, 2005
This review article discusses the reaction of nitrilimines and nitrile oxides with hydrazines, hydrazones, and oximes. Three reaction modes were observed.
Awadallah, Adel M., Ferwanah, Abdel-Rahman S.   +1 more
core   +2 more sources

A new convenient synthesis of 3-hetaryl-pyrazolo[5,1-c][1,2,4]triazines

Journal of Advanced Research, 2012
Reactions of enaminones 2 with diazotized 5-amino-3-phenylpyrazole provide a convenient route to 3-[(4,5-disubstituted-pyrazol-3-yl)carbonyl]-pyrazolo[5,1-c][1,2,4]triazines.
Ahmad S. Shawali
doaj   +1 more source

Chemistry of the Enaminone of 1-Acetylnaphthalene under Microwave Irradiation Using Chitosan as a Green Catalyst

Molecules, 2011
Enaminone 1 was reacted with hydrazonoyl halides 2a-d to yield 3,4-disubstituted pyrazoles 6a-d. Coupling with arenediazonium chlorides afforded the 2-(arylhydrazono)-3-(1-naphthalenyl)-3-oxopropionaldehydes 13a-c.
Huwaida M. E. Hassaneen
doaj   +1 more source

Synthesis and Antimicrobial Studies of Some Novel Bis-[1,3,4]thiadiazole and Bis-thiazole Pendant to Thieno[2,3-b]thiophene Moiety [PDF]

, 2012
The synthetic utility of 3,3′-(3,4-dimethylthieno[2,3-b]thiophene-2,5-diyl)bis (3-oxopropanenitrile) (1) in the synthesis of some novel bis-[1,3,4-thiadiazole] 6a–g and bis-thiazole 10 and 13 derivatives with thieno[2,3-b]thiophene moiety is reported ...
Kheder, Nabila Abdelshafy, Mabkhot, Yahia Nasser   +1 more
core   +3 more sources