Results 121 to 130 of about 1,345 (190)

Xanthene-to-fluorene skeletal editing <i>via</i> oxygen deletion mediated by boron and aluminium radicals. [PDF]

Chem Sci
Nahon E, Nelmes GR, Dallerba E, Lim LF, Cox N, McMullin CL, Massi M, Kallmeier F, Hicks J.   +8 more
europepmc   +1 more source

Electrochemical Synthesis of Unnatural Amino Acids Embedding 5- and 6-Membered Heteroaromatics. [PDF]

ACS Omega
Bombonato E, Fasano V, Pecorari D, Fornasari L, Castagnini F, Marcaccio M, Ronchi P.   +6 more
europepmc   +1 more source

Methylene Insertion into Nitrogen-Heteroatom Single Bonds of 1,2-Azoles via a Zinc Carbenoid: An Alternative Tool for Skeletal Editing. [PDF]

Adv Sci (Weinh)
Tsuda M, Morita T, Morita Y, Takaya J, Nakamura H.   +4 more
europepmc   +1 more source

Analysis of the structural diversity of heterocycles amongst European medicines agency approved pharmaceuticals (2014-2023). [PDF]

RSC Med Chem
Ward M, O'Boyle NM.
europepmc   +1 more source

Organophotocatalytic Functionalization of 3,4-Dihydroquinoxalin-2-ones with Isoxazol-5-amines Using Visible Light. [PDF]

J Org Chem
Mora-Rodríguez SE, Rostoll-Berenguer J, Lagunas S, Vázquez MA, Blay G, Pedro JR, Vila C.   +6 more
europepmc   +1 more source

Menaquinone depletion resensitises bedaquiline-resistant tuberculosis

Wetzel J, Dallow J, Davis E, Pearson WH, Daems S, Govaerts M, Hereijgers J, Sprangers J, Truebody B, Maes V, van Hasselt V, Leemans A, Pujari V, Vos A, Martínez Viturro CM, Enrique Gómez J, Peeters M, Gerber M, Chhabra N, Wouters A, Everaerts M, Painter H, Fathima R, Willcocks SJ, Davies C, Raeymaekers V, Clark TG, Draghia-Akli R, Fletcher H, Van Loock M, Hibberd ML, Mostowy S, Crick DC, Pym AS, Samby K, Jackson P, Trabanco AA, Larrouy-Maumus G, Steyn AJ, Stoops B, Dhar N, Aguilar-Pérez C, Lamprecht DA, Wall RJ, Koul A.   +44 more
europepmc   +1 more source

3-Chloro-4-(p-tolyl)isothiazole-5-carbonitrile

MolBank, 2023
A reaction of 3-chloroisothiazole-5-carbonitrile with 1-iodo-4-methylbenzene (2 equiv.) produced 3-chloro-4-(p-tolyl)isothiazole-5-carbonitrile in a 60% yield.
Panayiotis A Koutentis, Andreas S Kalogirou   +1 more
exaly   +2 more sources

Anti-HIV evaluation of benzo[d]isothiazole hydrazones

European Journal of Medicinal Chemistry, 2009
The synthesis and the anti-HIV-1 activity of novel benzo[d]isothiazole hydrazones are reported. Target compounds tested in MT-4 cells cultures for their anti-HIV properties against wild type HIV-1 and HIV strains carrying clinically relevant mutations ...
Roberta Loddo, Matteo Incerti, Paolo la Colla   +2 more
exaly   +2 more sources

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Isothiazoles

Angewandte Chemie International Edition in English, 1963
AbstractThe ring system of non‐anellated 1,2‐thiazoles (isothiazoles) has only recently become accessible. Four syntheses and numerous interconversions have opened up new routes to compounds which command interest as intermediates and as analogues of natural products and established pharmaceuticals.
F. Hübenett, H. D. Hofmann
openaire   +2 more sources

In Silico Exploration for Identifying Structure–Activity Relationship of MEK Inhibition and Oral Bioavailability for Isothiazole Derivatives [PDF]

Chemical Biology and Drug Design, 2010
In this study, quantitative structure–activity ⁄prop-erty models are developed for modeling and pre-dicting both MEK inhibitory activity and oral bioavailability of novel isothiazole-4-carboxami-dines.
Georgia Melagraki, Antreas Afantitis, Panayiotis A Koutentis   +2 more
exaly   +2 more sources