Results 81 to 90 of about 871 (158)

Methylene Insertion into Nitrogen-Heteroatom Single Bonds of 1,2-Azoles via a Zinc Carbenoid: An Alternative Tool for Skeletal Editing. [PDF]

Adv Sci (Weinh)
Tsuda M, Morita T, Morita Y, Takaya J, Nakamura H.   +4 more
europepmc   +1 more source

Organophotocatalytic Functionalization of 3,4-Dihydroquinoxalin-2-ones with Isoxazol-5-amines Using Visible Light. [PDF]

J Org Chem
Mora-Rodríguez SE, Rostoll-Berenguer J, Lagunas S, Vázquez MA, Blay G, Pedro JR, Vila C.   +6 more
europepmc   +1 more source

Analysis of the structural diversity of heterocycles amongst European medicines agency approved pharmaceuticals (2014-2023). [PDF]

RSC Med Chem
Ward M, O'Boyle NM.
europepmc   +1 more source

Reactions of acryl thioamides with iminoiodinanes as a one-step synthesis of <i>N</i>-sulfonyl-2,3-dihydro-1,2-thiazoles. [PDF]

Beilstein J Org Chem
Ilkin VG, Silaichev PS, Filimonov VO, Beryozkina TV, Likhacheva MD, Slepukhin PA, Dehaen W, Bakulev VA.   +7 more
europepmc   +1 more source

Synthesis and Biological Activity of Novel Polyazaheterocyclic Derivatives of Quinine. [PDF]

Molecules
Mukusheva GK, Toigambekova NN, Seidakhmetova RB, Jalmakhanbetova RI, Babakhanova MN, Nurkenov OA, Akishina EA, Dikusar EA, Kolesnik IA, Zhou H, Potkin VI.   +10 more
europepmc   +1 more source

Synthesis of a 3,7-Disubstituted Isothiazolo[4,3-b]pyridine as a Potential Inhibitor of Cyclin G-Associated Kinase. [PDF]

Molecules
Grisez T, Ravi NP, Froeyen M, Schols D, Van Meervelt L, De Jonghe S, Dehaen W.   +6 more
europepmc   +1 more source

EGFR Mutations and Tyrosine Kinase Inhibitors: Structural Insights and Therapeutic Advances. [PDF]

ACS Omega
Manoj MV, Mupparaju V RB, Thakur A, Sasidharan Pillai AK.   +3 more
europepmc   +1 more source

The Selective 3-MST Inhibitor I3MT-3 Works as a Potent Caspase-1 Inhibitor. [PDF]

Int J Mol Sci
Otani K, Komatsu R, Noguchi T, Suzuki W, Hirata Y, Matsuzawa A.   +5 more
europepmc   +1 more source

Semisynthesis of Mycothiazole Analogs having Distinct Bioactivity. [PDF]

ACS Med Chem Lett
Clarke JG, Dutta N, Nickel MS, Wang Z, Kim J, Media J, Coppage DA, McCauley EP, Gerke JA, Anderson MO, Higuchi-Sanabria R, Valeriote FA, Crews P, Johnson TA.   +13 more
europepmc   +1 more source

A patent review of von Hippel-Lindau (VHL)-recruiting chemical matter: E3 ligase ligands for PROTACs and targeted protein degradation (2019-present). [PDF]

Expert Opin Ther Pat
Urbina A, Hallatt AJ, Robertson J, Ciulli A.   +3 more
europepmc   +1 more source