Results 21 to 30 of about 8,655 (241)

Green Synthesis, Characterization, and Biochemical Impacts of New Bioactive Isoxazoline-sulfonamides as Potential Insecticidal Agents against the Sphodroxia Maroccana Ley.

Pest Management Science, 2023
BACKGROUND Sphodroxia maroccana Ley is a pest of cork oak crops that damages the roots of seedlings and can severely impair cork oak regeneration. Since the banning of carbosulfan and chlorpyriphos widely used against the larvae of Sphodroxia maroccana ...
Ayoub El Mahmoudi, R. Fegrouche, Hamza Tachallait, J. Lumaret, S. Arshad, K. Karrouchi, K. Bougrin   +6 more
semanticscholar   +1 more source

Development of Potent 3Br-isoxazoline-Based Antimalarial and Antileishmanial Compounds

, 2021
Starting from the structure of previously reported 3-Br-isoxazoline-based covalent inhibitors of P. falciparum glyceraldehyde 3-phosphate dehydrogenase, and with the intent to improve their metabolic stability and antimalarial activity, we designed and ...
Nicoletta Basilico (806898), Andrea Galbiati (6393374), Donatella Taramelli, Lucia Tamborini, Nicoletta Basilico, Aureliano Zana, Lucia Tamborini (810793), Consuelo Coser (11558679), Consuelo Coser, Paola Conti, Aureliano Zana (11558676), Andrea Galbiati, Paola Conti (810797), Silvia Parapini, Silvia Parapini (806899), Donatella Taramelli (736311)   +15 more
core   +1 more source

The mode of action of isocycloseram: A novel isoxazoline insecticide.

Pesticide Biochemistry and Physiology, 2022
Isocycloseram is a novel isoxazoline insecticide and acaricide with activity against lepidopteran, hemipteran, coleopteran, thysanopteran and dipteran pest species.
Judith Blythe, F. Earley, Katarzyna Piekarska-Hack, Lucy C. Firth, Julia Bristow, E. Hirst, James A. Goodchild, E. Hillesheim, Andrew J. Crossthwaite   +8 more
semanticscholar   +1 more source

New (S)-verbenone-isoxazoline-1,3,4-thiadiazole hybrids: synthesis, anticancer activity and apoptosis-inducing effect

, 2023
Background: This study aimed to develop novel isoxazoline-1,3,4-thiadiazole hybrids from (S)-verbenone for potential anticancer treatment, particularly focusing on cytotoxic and apoptotic effects in hormonesensitive MCF-7 and triple-negative MDA-MB-231 ...
Mourad Fawzi (10304096), El Mostafa Ketatni (17065748), Aziz Auhmani (10304105), Abdellah N’ait Oussidi (17065747), Hamid Morjani (27104), Lahcen EL Ammari (15379430), Abdoullah Bimoussa (12809505), Ali Oubella (10304090), Mohamed Saadi (755383), Yassine Laamari (10304099), Moulay Youssef Ait Itto (15996891)   +10 more
core   +1 more source

Synthesis of Functionalized 4,5-Dihydroisoxazoles Decorated with the Dimethylphosphinoyl Group

Журнал органічної та фармацевтичної хімії, 2023
Aim. To synthesize a hybrid molecular platform incorporating dimethylphosphinoyl and 4,5-dihydroisoxazole moieties suitable for the creation of focused combinatorial libraries of compounds. Results and discussion.
Andrii V. Fedyk, Bohdan A. Chalyk
doaj   +1 more source

Synthesis, Characterization, DFT Mechanistic Study, Antimicrobial Activity, Molecular Modeling, and ADMET Properties of Novel Pyrazole-isoxazoline Hybrids

ACS Omega, 2022
A series of new heterocycle hybrids incorporating pyrazole and isoxazoline rings was successfully synthesized, characterized, and evaluated for their antimicrobial responses.
Mohammed Chalkha, H. Nour, Khalid Chebbac, A. Nakkabi, Lahoucine Bahsis, Mohamed Bakhouch, Mohamed Akhazzane, M. Bourass, S. Chtita, Y. B. Bin Jardan, M. Augustyniak, Mohammed Bourhia, Mourad A. M. Aboul-Soud, M. el Yazidi   +13 more
semanticscholar   +1 more source

Toxicity and Sublethal Effects of Fluxametamide on the Key Biological Parameters and Life History Traits of Diamondback Moth Plutella xylostella (L.)

Agronomy, 2022
Fluxametamide, a novel isoxazoline insecticide, is newly registered for the control of various lepidopteran, coleopteran and thysanopteran insect pests on lethal and sublethal levels.
Amit Gope, Gautam Chakraborty, Shanowly Mondal Ghosh, Sayan Sau, Krishnendu Mondal, Abhisek Biswas, Sukamal Sarkar, Pijush Kanti Sarkar, Debashis Roy   +8 more
doaj   +1 more source

Current review of isoxazoline ectoparasiticides used in veterinary medicine.

Journal of Veterinary Pharmacology and Therapeutics, 2021
The isoxazolines are a novel class of ectoparasiticides with potent inhibitory activity on glutamate- and gamma-aminobutyric acid-gated chloride channel located in nervous system of invertebrates.
Xueying Zhou, A. Hohman, W. Hsu
semanticscholar   +1 more source

3′,4′-Diphenyl-3H,4′H-spiro[benzo[b]thiophene-2,5′-isoxazol]-3-one

IUCrData, 2018
The molecule of the title compound, C22H15NO2S, is built up from a benzothiophene system linked to an isoxazoline ring which is connected to two phenyl rings.
Mohamed Bakhouch, Mohamed El Yazidi, Ghali Al Houari, Mohamed Saadi, Lahcen El Ammari   +4 more
doaj   +1 more source

Electrochemical Synthesis of Isoxazolines: Method and Mechanism [PDF]

Chemistry – A European Journal, 2022
Abstract An electrochemical method for the green and practical synthesis of a broad range of substituted isoxazoline cores is presented. Both aryl and more challenging alkyl aldoximes are converted to the desired isoxazoline in an electrochemically enabled regio‐ and diastereoselective reaction with electron‐deficient alkenes ...
Holman, Samuel D. L., Wills, Alfie G., Fazakerley, Neal J., Poole, Darren L., Coe, Diane M., Berlouis, Leonard, Reid, Marc   +6 more
openaire   +5 more sources