Beilstein Journal of Organic Chemistry, 2018 Hypervalent iodine-mediated olefin functionalization provides a rapid gateway towards accessing both various heterocyclic cores and functional groups.
Sang Won Park +6 more
doaj +3 more sources
Synthesis and Pharmacological Significance of Isoxazoline Derivatives: A Mini review [PDF]
Academic Science JournalFive-membered heterocycles, like isoxazolines, are an important class of compounds of bioorganic and pharmacological importance. They have been treated as useful intermediates for the transformation of a large number of bioactive molecules.
mohammed alwan
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Synthesis and antibacterial studies of some novel isoxazoline derivatives [PDF]
Journal of the Serbian Chemical Society, 2007 A series of 3-[3-(2,4-dichloro-5-fluorophenyl)-5-(2-furyl)-4,5-dihydro-1H-pyrazol-1-yl]-5-(substituted phenyl/2-thienyl)isoxazolines (4a-j) were prepared. The structures of the isoxazoline derivatives were confirmed on the bases of elemental analysis and
TEJASKUMAR SHAH, VIKAS DESAI
doaj +4 more sources
The mosquitocidal activity of isoxazoline derivatives afoxolaner, lotilaner, and fluralaner are not affected by mosquito sugar or antibiotic treatment [PDF]
Scientific ReportsLong-lasting insecticidal nets and indoor residual sprays have played a major role in significantly reducing the burden of malaria. However, the management of mosquitoes resistant to current insecticides continues to be challenging.
Harouna Soré +8 more
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Asymmetric Synthesis of Functionalized 2-Isoxazolines. [PDF]
ACS OmegaThe asymmetric synthesis of the isoxazoline skeleton was achieved by the oxidation of hydroxylaminoalkyl furan prepared from simple starting materials: 2-methylfuran and (S)-epichlorohydrin. The synthesis features an NBS-mediated oxidation of hydroxylaminoalkyl furan to give an α,β-unsaturated ketone intermediate which cyclized to the isoxazoline.
Hamur B +5 more
europepmc +4 more sources
Renewed «Isoxazoline Route» for the Synthesis of Densely Functionalized Ketones [PDF]
, 2022 In this work, the «isoxazoline route» to aldols involving the [3+2]-cycloaddition of nitrile oxide to alkenes and hydrogenolysis of oxime group was revisited.
Pavel, Ushakov +2 more
core +1 more source
Synthesis, DFT Study and Antibacterial Activity of some Isoxazoline Derivatives Containing 1,4-benzothiazin-3-one Nucleus Obtained Using 1,3-dipolar Cycloaddition Reaction [PDF]
Iranian Journal of Chemistry & Chemical Engineering, 2020 Novel series of isoxazoline derivatives containing 1,4-benzothiazin-3-one ring (6a-h) were synthesized via 1,3-dipolar cycloaddition reactions of arylnitrile oxides 5a-d on 4-allyl-2-(substituted)-1,4-benzothiazin-3-ones 3 and 4 led to polyheterocyclic ...
Sebbar Nada Kheira +8 more
doaj +1 more source
An easy access to chromano-isoxazolines and functionalized isoxazolines [PDF]
Arkivoc, 2004 2-Allyloxybenzaldoximes on treatment with ceric ammonium nitrate (CAN) at room temperature afforded 3a,4-dihydro-3H-chromeno[4,3-c]isoxazoles while benzaldoximes on interaction with Baylis-Hillman adduct in the presence of CAN produced functionalized isoxazolines.
Biswanath Das +3 more
openaire +1 more source
Toxics, 2023 The fall armyworm (FAW), Spodoptera frugiperda, is one of the most devastating invasive polyphagous pests, which has attracted recent global attention by developing resistance to various insecticidal active ingredients with independent mode of action ...
Debashis Roy +9 more
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The Potential of Fluralaner as a Bait Toxicant to Control Pest Yellowjackets in California
Insects, 2023 The western yellowjacket, Vespula pensylvanica (Saussure), is an important seasonal pest of recreational and outdoor venues in the western United States. Its propensity to scavenge food increases the likelihood of stinging incidences.
Michael K. Rust +11 more
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