VARIOUS BIOLOGICAL ACTIVITIES OF COUMARIN AND OXADIAZOLE DERIVATIVES [PDF]
In this review article data is collected regarding the various derivatives of coumarin and oxadiazole as both these have wide range of biological activities and they can be further modified to synthesize more effective and potent drugs. Coumarin class of
Saini, Rupinder +4 more
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Synthesis and Synthetic Applications of 1,2,4-Oxadiazole-4-Oxides [PDF]
The first 1,2,4-oxadiazole-4-oxide was prepared by Wieland a century ago, but-this compound remained largely a chemical curiosity until very recently.
CARAMELLA, PIERLUIGI, QUADRELLI, PAOLO
core
A series of new 1,2,4-oxadiazole-based derivatives were synthesized and evaluated for their anti-AD potential. The results revealed that eleven compounds (1b, 2a-c, 3b, 4a-c, and 5a-c) exhibited excellent inhibitory potential against AChE, with IC50 ...
Mohammed Salah Ayoup +8 more
doaj +1 more source
A mini review on pharmacological activities of oxadiazole and thiadiazole compounds [PDF]
In the last few years, heterocyclic compounds have attracted strong interest and a lot of work has been done on oxadiazole and thiadiazole ring. Oxadiazole and thiadiazole a five member heterocyclic nucleus has attracted a wide attention of the chemist ...
Asif, Mohammad
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biological Aspects of 1,3,4 -oxadiazole derivatives [PDF]
Heterocyclic compounds analog have attracted wide attention due to their useful biological properties. Among them, 1,3,4-oxadiazoles have exhibiteda wide range of biological properties including anti-bacterial, anti-viral, anti-fungal, anti-cancer, anti ...
S, GNANAVEL, S, KAVITHA, K, KANNAN
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Oxadiazole carboxamide nucleosides as probes for DNA polymerases [PDF]
Azole carboxamide nucleosides represent a unique class of analogs that possess distinct electronic properties and structural versatility through the rotation of glycosidic and carboxamide bonds.
Adelfinskaya, Olga V
core
Design, synthesis, and enzyme kinetic evaluation of oxadiazole derivatives as nucleoside triphosphate diphosphohydrolase (NTPDase) inhibitors: an integrated <i>in vitro</i> and <i>in silico</i> approach. [PDF]
Abbas SZ +6 more
europepmc +1 more source
Multifunctional pectin derivatives as anticancer agents in colorectal cancer via synthesis, computational insights, and modulation of NRF2/HO-1, HIF-1α, and VEGF/PDGF-D signaling pathways. [PDF]
Elsayed GH, Fahim AM.
europepmc +1 more source
Benzo[<i>d</i>]imidazole anchored oxadiazole derivatives: synthesis, characterization, biological evaluation, <i>in silico</i> docking and ADME-T analysis. [PDF]
Salluri YR, Chepuri K, Anwar S.
europepmc +1 more source

