Recent Developments in Ferulic Acid- and Caffeic Acid-Based Hybrids with Potential Anticancer Properties. [PDF]
Peter S, Sibali LL, Khwaza V, Paca AM.
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A mini review on pharmacological activities of oxadiazole and thiadiazole compounds
In the last few years, heterocyclic compounds have attracted strong interest and a lot of work has been done on oxadiazole and thiadiazole ring. Oxadiazole and thiadiazole a five member heterocyclic nucleus has attracted a wide attention of the chemist ...
Asif, Mohammad
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Design, synthesis and antiproliferative, apoptotic, and immunomodulatory properties of new heteroaryl pyridine-linked 1,2,4-oxadiazoles as prospective dual EGFR/BRAF<sup>V600E</sup> inhibitors. [PDF]
Gomaa HAM +9 more
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biological Aspects of 1,3,4 -oxadiazole derivatives
Heterocyclic compounds analog have attracted wide attention due to their useful biological properties. Among them, 1,3,4-oxadiazoles have exhibiteda wide range of biological properties including anti-bacterial, anti-viral, anti-fungal, anti-cancer, anti ...
S, GNANAVEL, S, KAVITHA, K, KANNAN
core
Novel pyrazole-oxadiazole-chalcone/oxime hybrids as dual EGFR/VEGFR-2 inhibitors with promising anticancer potential: a comprehensive cytotoxicity evaluation, mechanistic insights and SAR analysis. [PDF]
Alshazly O +3 more
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Oxadiazole carboxamide nucleosides as probes for DNA polymerases
Azole carboxamide nucleosides represent a unique class of analogs that possess distinct electronic properties and structural versatility through the rotation of glycosidic and carboxamide bonds.
Adelfinskaya, Olga V
core
Lonidamine-1,3,4-oxadiazole derivatives with antiproliferative effects on HCT116 colon cancer cell lines: biological evaluation, ADMET, and computational studies. [PDF]
Bhat RM +6 more
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Bridging mechanism and design: modern medicinal chemistry approaches to thymidylate synthase inhibitors. [PDF]
Al-Karmalawy AA +4 more
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Design, synthesis and antiproliferative activity of oxadiazole derivatives as potent glycogen synthase kinase-3/histone deacetylase 6 dual inhibitors. [PDF]
Ye C +7 more
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Exploring 1,3,4-oxadiazolyl sulfide derivatives as antidiabetic candidates: synthesis, antioxidant activity, SAR-study, molecular docking, and DFT-insights. [PDF]
Khalaf NA +3 more
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