Results 151 to 160 of about 12,035 (216)

Novel Imidazopyridine-Oxadiazole β‑Tubulin Inhibitors Suppress Breast Cancer Migration and Induce Caspase-3-Mediated Apoptosis. [PDF]

ACS Omega
Cakir M, Kuzu B.
europepmc   +1 more source

Bis-Oxadiazole Assemblies as NO-Releasing Anticancer Agents. [PDF]

Pharmaceutics
Matnurov EM, Stebletsova IA, Larin AA, Arakelyan J, Ananyev IV, Gushchin AL, Fershtat LL, Babak MV.   +7 more
europepmc   +1 more source

Water-Soluble Heptacyclic Oligo-Heteroaryls Targeting G‑Quadruplex DNA via Groove-Binding Interactions. [PDF]

ACS Omega
Fracchioni G, Caramiello AM, Nadai M, Lena A, Freccero M, Richter SN, Pirota V, Doria F.   +7 more
europepmc   +1 more source

Novel Isoniazid-Based 1,3,4-Oxadiazole-Fatty Acid Hybrids: Synthesis, In Vitro Biological Activity and In Silico ADME/Tox Predictions. [PDF]

Chem Biodivers
Jadhaw B, Kumar CB, Vasapalli K, Pranathi KS, Ramesh G, Misra S, Kaki SS.   +6 more
europepmc   +1 more source

Lead Optimization: Synthesis and Biological Evaluation of Griseofulvin Derivatives as Novel SIRT6 Activators. [PDF]

ACS Med Chem Lett
Zorko T, Kogovšek J, Ciber L, Ostojić I, Maraš N, Novinec M, Štefane B.   +6 more
europepmc   +1 more source

A two-decade overview of oxadiazole derivatives as promising anticancer agents. [PDF]

RSC Adv
Salem M, El-Adl K, El-Morsy A, Abulkhair HS.   +3 more
europepmc   +1 more source

Integrating Experimental Physicochemical Data with PBPK Modeling to Guide the Translational Development of the Antifungal 1,3,4-Oxadiazole Derivative LMM6. [PDF]

ACS Omega
Piai JMB, Lippa VNM, Caleffi-Marchesini ER, Borghi Pangoni FB, Felipe MS, Kioshima ES, Diniz A.   +6 more
europepmc   +1 more source

Novel 1,2,4-Oxadiazole Derivatives in Drug Discovery

Pharmaceuticals, 2020
Five-membered 1,2,4-oxadiazole heterocyclic ring has received considerable attention because of its unique bioisosteric properties and an unusually wide spectrum of biological activities.
Janusz Rachon, Konrad Kubiński, Mateusz Dasko   +2 more
exaly   +2 more sources

Synthesis and antimicrobial activity of some 1,3,4-oxadiazole derivatives

Il Farmaco, 2002
Six new 5-(1-/2-naphthyloxymethyl)-1,3,4-oxadiazole-2(3H)-thione, 2-amino-5-(1-/2-naphthyloxymethyl)-1,3,4-oxadiazole, 5-(1-/ 2-naphthyloxymethyl)-1,3,4-oxadiazole-2(3H)-one derivatives have been synthesized from 1-and/or 2-naphthol.
Melike Ekizoğlu, Erhan Palaska, Meral Özalp   +2 more
exaly   +2 more sources