Results 121 to 130 of about 17,763 (235)

Evidence of an activity-enhancing conformational shift in Arabidopsis thaliana plant cysteine oxidase 4 induced by binding of substrate or substrate-mimics. [PDF]

J Biol Chem
Latter R, Hintzen JCJ, Shah LMN, Gunawardana DM, Sher RM, White MD, Mecinović J, Benesch JLP, Flashman E.   +8 more
europepmc   +1 more source

Peptidomimetic Modified Heptamethine Cyanine Dyes for Enhanced Bioimaging Targetability: A Molecular Interaction Study on Bovine Serum Albumin and Human Parvalbumin. [PDF]

J Med Chem
Ahmed TE, Azizi-Khereshki N, Henary M.
europepmc   +1 more source

Deconvolution of the On-Target Activity of Plasmepsin V Peptidomimetics in <i>Plasmodium falciparum</i> Parasites. [PDF]

ACS Infect Dis
Su W, Nguyen W, Siddiqui G, Dziekan JM, Marapana D, Penington JS, Mehra S, Razook Z, McCann K, Ngo A, Jarman KE, Barry AE, Papenfuss AT, Gilson PR, Creek DJ, Cowman AF, Sleebs BE, Dans MG.   +17 more
europepmc   +1 more source

Retraction Note: Thiazole-valine peptidomimetic (TTT-28) antagonizes multidrug resistance in vitro and in vivo by selectively inhibiting the efflux activity of ABCB1. [PDF]

Sci Rep
Wang YJ, Patel BA, Anreddy N, Zhang YK, Zhang GN, Alqahtani S, Singh S, Shukla S, Kaddoumi A, Ambudkar SV, Talele TT, Chen ZS.   +11 more
europepmc   +1 more source

On-Resin Synthesis and Diversification of Macrocyclic Disulfide Bridge Peptidomimetics via Bifunctional 5-Iodo-1,4-Triazoles. [PDF]

J Org Chem
Malone MA, Shepperson OA, Simms JE, Reid AJ, Jamieson AG.   +4 more
europepmc   +1 more source

Next-generation inhibitors of SARS-CoV-2 M^pro overcome the deficiencies of Paxlovid. [PDF]

Nat Commun
Luo G, Wang G, Liao C, Zhong B, Fan L, Zhang J, Rao J, Zhang J, Wang Z, Luo M, Yan Y, Lu L, Xu W, Wu F, Gao X, Lu W.   +15 more
europepmc   +1 more source

Design and In Vitro Evaluation of Novel GC373-like SARS-CoV-2 Main Protease Inhibitors. [PDF]

Curr Issues Mol Biol
Kuznetsova AA, Makhin AP, Bulygin AA, Andrianova AA, Miturich VS, Zagitova RI, Shmygarev VI, Fadeeva AA, Yatskin ON, Belozerova OA, Smirnov IV, Yampolsky IV, Kaskova ZM, Kuznetsov NA.   +13 more
europepmc   +1 more source

Role of Structural Modifications in Peptidomimetic Compounds as Potential Antimicrobial Agents against <i>Staphylococcus aureus</i> and <i>Streptococcus pyogenes</i>: Balancing Bioavailability, Safety, and Antimicrobial Activity. [PDF]

ACS Omega
Dzierżyńska M, Sawicka J, Łada K, Gajewicz-Skretna A, Deptuła M, Chernobrovkin A, Pogorzelska A, Grubb A, Zubarev RA, Pikuła M, Kasprzykowski F, Rodziewicz-Motowidło S.   +11 more
europepmc   +1 more source

Novel macrocyclic peptidomimetics targeting the insulin-regulated aminopeptidase (IRAP): design, synthesis and evaluation. [PDF]

RSC Med Chem
Olaniran Håkansson E, Balestri LJI, Puthiyaparambath S, Moes S, Henschel H, Sköld C, Hallberg M, Larhed M, Skillinghaug B, Odell LR.   +9 more
europepmc   +1 more source

High-Affinity Peptidomimetic Inhibitors of the DCN1-UBC12 Protein-Protein Interaction.

Journal of Medicinal Chemistry, 2018
Haibin Zhou, Weihua Zhou, Bing Zhou, Liu Liu, Ting‐Rong Chern, Krishnapriya Chinnaswamy, Jianfeng Lu, D. Bernard, Chao-Yie Yang, Shasha Li, Mi Wang, J. Stuckey, Yi Sun, Shaomeng Wang   +13 more
semanticscholar   +1 more source