Results 141 to 150 of about 17,763 (235)

A Three-Layer Transformation Strategy toward Functionalized Fused Hydantoins and Diketopiperazines. [PDF]

Org Lett
Giannakaki MA, Zingiridis M, Froudas KG, Neochoritis CG.   +3 more
europepmc   +1 more source

Structural basis of TMPRSS11D specificity and autocleavage activation. [PDF]

Nat Commun
Fraser BJ, Wilson RP, Ferková S, Ilyassov O, Lac J, Dong A, Li YY, Seitova A, Li Y, Hejazi Z, Kenney TMG, Penn LZ, Edwards A, Leduc R, Boudreault PL, Morin GB, Bénard F, Arrowsmith CH.   +17 more
europepmc   +1 more source

Covalent Radiopharmaceuticals: Precision Imaging and Therapy for Cancer. [PDF]

Mol Pharm
Klauser PC, Wang L.
europepmc   +1 more source

Covalent Peptide-Based N-Myc/Aurora-A Inhibitors Bearing Sulfonyl Fluoride Warheads. [PDF]

J Pept Sci
Dawber RS, Gimenez D, Preston GW, Wright MH, Bayliss R, Warriner SL, Wilson AJ.   +6 more
europepmc   +1 more source

Inhibition of Human Coronavirus 229E by Lactoferrin-Derived Peptidomimetics. [PDF]

Pharmaceutics
Scala MC, Marchetti M, Landi M, Fantacuzzi M, Superti F, Agamennone M, Campiglia P, Sala M.   +7 more
europepmc   +1 more source

Nano-G_s Protein Peptidomimetics: Rational Design of Gα C-Terminus-Derived Peptides Mimicking Key Components of G_s-β₂AR Interactions. [PDF]

Angew Chem Int Ed Engl
Tran PT, Danielsen M, Tiemann JKS, Ibrahim P, Rasmussen SGF, Kubiak X, Batebi H, Gadais C, Ballet S, Hildebrand PW, Pedersen DS, Mathiesen JM.   +11 more
europepmc   +1 more source

Thiazole peptidomimetics as chemical modulators of <i>KRAS</i> gene expression <i>via</i> G-quadruplex stabilization. [PDF]

RSC Chem Biol
Biswas D, Gorai A, Maiti S, Chaudhuri R, Pradhan S, Dash J.   +5 more
europepmc   +1 more source

Fat or flat? The impact of dipole moment vectors on non-covalent interactions between aromatic tags and macromolecules.

Inorg Chem Front
Holub J, Jílková A, Lemke C, Cianni L, Spiwoková P, Horn M, Breuer C, Leontovyč A, Brynda J, Mertlíková-Kaiserová H, Chanová M, Dos Reis Rocho F, Montanari CA, El-Sakkary N, Caffrey CR, Gütschow M, Hnyk D, Mareš M, Fanfrlík J.   +18 more
europepmc   +1 more source

Advancements in development of novel class of HIV protease inhibitors. [PDF]

Ann Med
Gu WG, Yin GZ, Zhang YP.
europepmc   +1 more source

Native MS and ligand observed NMR uncovers subtle SLiM binding variations that mediate HSP90-Hop PPI modulation. [PDF]

RSC Chem Biol
Davids TK, Kusza DA, Misplon SK, Späth JC, Mhlanga R, Clarke DJ, de la Torre BG, Albericio F, Edkins AL, Rylands M, Veale CGL.   +10 more
europepmc   +1 more source