Results 141 to 150 of about 14,095 (224)

<i>N</i>‑Acyl Hemiperaminals: From Bioactive Skeleton Editing of Artemisinin to Programmable Handles for α‑Amido Functionalization and Bioactive Peroxides. [PDF]

JACS Au
Li Y, Gao H, Ye J, Zhou H, Zhu Q, Rao D, Li L, Wang L, Zuo D, Lin T, Wang S, Deng X, Zheng X.   +12 more
europepmc   +1 more source

Recent Exploration of Right-Handed D-Sulfonyl-γ-AApeptides as Potential Tools Toward α-Helical Mimicry. [PDF]

Chempluschem
Fontaine J, Cai J.
europepmc   +1 more source

BamA as a next-generation antibacterial target: mechanistic insights, inhibitor landscape, and rational drug design strategies. [PDF]

RSC Adv
Al-Karmalawy AA, Al Khatib AO, Hawas SS.
europepmc   +1 more source

Access to Cyclic Monensin Derivatives via a Four-Component Ugi Reaction. [PDF]

J Org Chem
Graniczny R, Huczyński A, Janczak J, Kłopotowska D, Wietrzyk J, Sulik M.   +5 more
europepmc   +1 more source

Retraction Note: Thiazole-valine peptidomimetic (TTT-28) antagonizes multidrug resistance in vitro and in vivo by selectively inhibiting the efflux activity of ABCB1. [PDF]

Sci Rep
Wang YJ, Patel BA, Anreddy N, Zhang YK, Zhang GN, Alqahtani S, Singh S, Shukla S, Kaddoumi A, Ambudkar SV, Talele TT, Chen ZS.   +11 more
europepmc   +1 more source

Enhanced antinociception of mixed efficacy opioid peptidomimetics through P-glycoprotein modulation. [PDF]

J Pharmacol Exp Ther
Anand JP, Kochan KE, Montgomery D, Nastase AF, Mosberg HI, Jutkiewicz EM.   +5 more
europepmc   +1 more source

On-Resin Synthesis and Diversification of Macrocyclic Disulfide Bridge Peptidomimetics via Bifunctional 5-Iodo-1,4-Triazoles. [PDF]

J Org Chem
Malone MA, Shepperson OA, Simms JE, Reid AJ, Jamieson AG.   +4 more
europepmc   +1 more source

Next-generation inhibitors of SARS-CoV-2 M^pro overcome the deficiencies of Paxlovid. [PDF]

Nat Commun
Luo G, Wang G, Liao C, Zhong B, Fan L, Zhang J, Rao J, Zhang J, Wang Z, Luo M, Yan Y, Lu L, Xu W, Wu F, Gao X, Lu W.   +15 more
europepmc   +1 more source

Opioid Peptide Hybrids as Multifunctional Analgesic Ligands: Emphasis on Intracellular Signaling. [PDF]

Pharmaceuticals (Basel)
Cecherz I, Waśkiewicz J, Dudek A, Polatyński D, Wtorek K, Piekielna-Ciesielska J.   +5 more
europepmc   +1 more source

Design and In Vitro Evaluation of Novel GC373-like SARS-CoV-2 Main Protease Inhibitors. [PDF]

Curr Issues Mol Biol
Kuznetsova AA, Makhin AP, Bulygin AA, Andrianova AA, Miturich VS, Zagitova RI, Shmygarev VI, Fadeeva AA, Yatskin ON, Belozerova OA, Smirnov IV, Yampolsky IV, Kaskova ZM, Kuznetsov NA.   +13 more
europepmc   +1 more source