Results 191 to 200 of about 26,717 (273)

Development of ketobenzothiazole-based peptidomimetic TMPRSS13 inhibitors with low nanomolar potency. [PDF]

J Enzyme Inhib Med Chem
Joushomme A, Désilets A, Champagne W, Hassanzadeh M, Lemieux G, Gravel-Trudeau A, Lepage M, Lafrenière S, Froehlich U, List K, Boudreault PL, Leduc R.   +11 more
europepmc   +1 more source

Epigenetic reader chromodomain as a potential therapeutic target. [PDF]

RSC Chem Biol
Sharma S, Hampton JT, Kutateladze TG, Liu WR.   +3 more
europepmc   +1 more source

Antinociceptive effects of intrathecal neuropeptide B/W receptor 1 agonists in mouse acute nociception, peripheral neuropathy, and inflammatory pain models. [PDF]

Pharmacol Rep
Ortiz YT, Nguyen T, Wilkerson JL.
europepmc   +1 more source

Stereoslektive Synthese von Prolin-Prolin-Dipeptidmimetika [PDF]

, 2011
Huy, Peter
core  

Rational design of small-sized peptidomimetic inhibitors disrupting protein-protein interaction. [PDF]

RSC Med Chem
Wang J, Zheng P, Yu J, Yang X, Zhang J.
europepmc   +1 more source

Rationally Designed Peptidomimetics

Proceedings of the 35th European Peptide Symposium, 2018
openaire   +1 more source

TMPRSS2 inhibitors with broad-spectrum efficacy against SARS-CoV-2 (JN.1) and influenza A (H1N1) viruses protect mice from influenza A infection. [PDF]

Emerg Microbes Infect
Presley L, Pérez-Vargas J, Saintigny A, Villanueva I, Ho M, Fone J, Brinsden L, Kaushik N, Olver S, Thompson CAH, Bautista-Sánchez D, Ennis S, Chen M, McCallum M, Brown JT, Ferková S, Hetrick B, Veesler D, Leduc R, Niikura M, Boudreault PL, Warner B, Jean F.   +22 more
europepmc   +1 more source

Synthesis, Antimicrobial Activity, and Tyrosinase Inhibition by Multifunctional 3,4-Dihydroxy-Phenyl Peptidomimetics. [PDF]

Int J Mol Sci
Wavhal DS, Koszelewski D, Kowalczyk P, Brodzka A, Ostaszewski R.   +4 more
europepmc   +1 more source

Evaluation of Cooperative Binding of Histone Post-Translational Modifications and the Surrounding Sequence by Trimethyllysine Reader Proteins. [PDF]

Biochemistry
Travis CR, Albanese KI, Henriksen HC, Kean KM, Waters ML.   +4 more
europepmc   +1 more source

Stapled histone H3 tails are super-substrates for lysine methyltransferase SETD7. [PDF]

Chem Sci
Bilgin N, Moesgaard L, Kongsted J, Mecinović J.   +3 more
europepmc   +1 more source