Results 111 to 120 of about 11,685 (174)

Therapeutic potential and safety challenges of antimicrobial peptides and peptidomimetics against ESKAPEE pathogens: a systematic review with quantitative analysis. [PDF]

J Antimicrob Chemother
Mekonen ES, Mishra SK, Urmi UL, Yeshtila YM, Maulvi FA, Kumar N, Willcox MDP.   +6 more
europepmc   +1 more source

Beyond Simple Mimicry: Next-Generation Geometric Architectures and Future Paradigms in Small-Molecule and Macrocyclic Peptidomimetics. [PDF]

Angew Chem Int Ed Engl
Lee J, Son S, Yoo JY, Lee JH, Chun M, Park SB.   +5 more
europepmc   +1 more source

Bilayer Permeabilization and the 'Sand-in-a-Gearbox' Mechanism for Membrane-Active Molecules: Which Is Which? [PDF]

Antibiotics (Basel)
Vaezi Z, Bortolotti A, Di Stefano C, Bonacorsi S, Santucci V, Carneri F, Aisenbrey C, Konai MM, Acharya Y, Venanzi M, Khosravi-Far R, Bechinger B, Haldar J, Stella L, Roversi D, Bocchinfuso G.   +15 more
europepmc   +1 more source

Recent Exploration of Right-Handed D-Sulfonyl-γ-AApeptides as Potential Tools Toward α-Helical Mimicry. [PDF]

Chempluschem
Fontaine J, Cai J.
europepmc   +1 more source

Beyond proteolysis: rational modification of mucin-derived peptidomimetics with enhanced metal-mediated antimicrobial activity. [PDF]

RSC Adv
Ślusarczyk A, Bellotti D, Leveraro S, Janek T, Zobi F, Remelli M, Wątły J.   +6 more
europepmc   +1 more source

Enhanced antinociception of mixed efficacy opioid peptidomimetics through P-glycoprotein modulation. [PDF]

J Pharmacol Exp Ther
Anand JP, Kochan KE, Montgomery D, Nastase AF, Mosberg HI, Jutkiewicz EM.   +5 more
europepmc   +1 more source

Extracellularly Activatable Conjugates of RGD Peptidomimetics and Cryptophycin for α_Vβ₃-Targeted Cancer Therapy. [PDF]

Chemistry
Seißenschmidt D, Hartung H, Kammer J, Sewald N.   +3 more
europepmc   +1 more source

Discovery of novel peptidomimetics against HSP90-HOP interactions towards improved cancer therapeutics using machine learning strategies. [PDF]

Front Bioinform
Perumal S, Karuppasamy R.
europepmc   +1 more source

On-Resin Synthesis and Diversification of Macrocyclic Disulfide Bridge Peptidomimetics via Bifunctional 5-Iodo-1,4-Triazoles. [PDF]

J Org Chem
Malone MA, Shepperson OA, Simms JE, Reid AJ, Jamieson AG.   +4 more
europepmc   +1 more source

Disrupting the Undruggable: Emerging Modalities for Targeting Protein-Protein Interactions in Oncology. [PDF]

Biology (Basel)
El-Tanani M, Rabbani SA, Wali AF, El-Tanani Y, Sharma S.   +4 more
europepmc   +1 more source