Results 91 to 100 of about 6,642 (186)

Covalent Peptide-Based N-Myc/Aurora-A Inhibitors Bearing Sulfonyl Fluoride Warheads. [PDF]

J Pept Sci
Dawber RS, Gimenez D, Preston GW, Wright MH, Bayliss R, Warriner SL, Wilson AJ.   +6 more
europepmc   +1 more source

Covalent Radiopharmaceuticals: Precision Imaging and Therapy for Cancer. [PDF]

Mol Pharm
Klauser PC, Wang L.
europepmc   +1 more source

GPepT: A Foundation Language Model for Peptidomimetics Incorporating Noncanonical Amino Acids. [PDF]

ACS Med Chem Lett
Oikawa Y, Uzawa T, Berenger F, Minagawa N, Yumoto A, Takaku H, Tamura R, Ito Y, Tsuda K.   +8 more
europepmc   +1 more source

Using generative AI to transform peptide hits into small molecule leads. [PDF]

Beilstein J Org Chem
Mills J, Lau YH.
europepmc   +1 more source

Antimicrobial activity of a short guanidine mimic immobilised on contact lenses. [PDF]

J Mater Sci Mater Med
Sara M, Kuppusamy R, Enninful G, Suresh D, Vasilev K, Mackenzie D, Dehghani F, Hui A, Wong EHH, Yasir M, Kumar N, Willcox M.   +11 more
europepmc   +1 more source

Antimicrobial nanocoatings and films for contact lenses: progress and promise. [PDF]

Nanomedicine (Lond)
Sara M, Attard S, Kumar N, Willcox M.
europepmc   +1 more source

Deconvolution of the On-Target Activity of Plasmepsin V Peptidomimetics in <i>Plasmodium falciparum</i> Parasites. [PDF]

ACS Infect Dis
Su W, Nguyen W, Siddiqui G, Dziekan JM, Marapana D, Penington JS, Mehra S, Razook Z, McCann K, Ngo A, Jarman KE, Barry AE, Papenfuss AT, Gilson PR, Creek DJ, Cowman AF, Sleebs BE, Dans MG.   +17 more
europepmc   +1 more source

Systematic Evaluation of Peptidomimetic Modifications in a Major Histocompatibility Complex Class I Model Epitope: A Framework for Immunogenic Antigen Design. [PDF]

ACS Chem Biol
Newkirk SE, Kelly JJ, Hourn N, Bhandari S, Spencer N, Pires MM.   +5 more
europepmc   +1 more source

Bridging Heterocycle-Mediated Hydrogen Bonding Facilitates Permeability of Polar Macrobicycles. [PDF]

J Am Chem Soc
Cooper GID, Dai B, Durham N, Walker GL, Yu H, Mendoza A, Bernardino SJ, Wu YD, Harran PG.   +8 more
europepmc   +1 more source

Opioid Affinity of Diazacyclic Peptidomimetic Compounds Derived from Reduced Polyamides. [PDF]

Int J Mol Sci
Chaudhari P, Bunnell A, Yegambaram M, Dooley C, Nefzi A.   +4 more
europepmc   +1 more source