Results 41 to 50 of about 11,685 (174)
Agonistic and antagonistic activities of the peptidomimetics against BdNTLR.
Agonistic and antagonistic activities of the peptidomimetics against BdNTLR.
Krzysztof Kaczmarek (3057564) +8 more
core +1 more source
Visualized and Quantitative Conformational Analysis of Peptidomimetics
Protein–protein interactions (PPIs) are fundamentally important and challenging drug targets. Peptidomimetic molecules of various types have been developed to modulate PPIs.
Hajime Takashima +15 more
core +1 more source
The synthesis of quinoline-based drugs has significant interest from researchers due to their broad spectrum of biological activities. In this context, a concise approach for the synthesis of quinoline-functionalized hybrid peptidomimetics is described ...
K. Ramya +5 more
doaj +1 more source
Development of Peptide Biopharmaceuticals in Russia
Peptides are low-molecular-weight substances that participate in numerous important physiological functions, such as human growth and development, stress, regulation of the emotional state, sexual behavior, and immune responses.
Vladislav I. Deigin +4 more
doaj +1 more source
Structure of the 4 peptidomimetics designed and synthesized.
Structure of the 4 peptidomimetics designed and synthesized.
Rong Chen (29176) +9 more
core +1 more source
Venom peptides and peptidomimetics as therapeutics
In the last 10 years, antimicrobial resistance (AMR) has become a huge public health concern with an estimated 10 million deaths per year and a projected $100 trillion impact on global the economy.
Ahmad, Zulfiqar, Akhtar, Suhail
core +1 more source
Despite the large number of peptidomimetics with incorporated heteroannularly functionalized ferrocenes, few studies have investigated their bioactivity.
Monika Kovačević +10 more
doaj +1 more source
Synthesis and Application of Triazole Containing Peptidomimetics [PDF]
Kracker O. Synthesis and Application of Triazole Containing Peptidomimetics.
Kracker, Oliver
core
Synthesis of Constrained Peptidomimetics via the Pictet-Spengler Reaction
Peptidomimetics offers a solution to the poor pharmacokinetic properties displayed by natural peptides, by providing pharmaceutically useful chemical structures with the ability to mimic the endogenous polyamide structure.
Vitaly V. Komnatnyy +5 more
core +1 more source
The nonstructural (NS) protein NS3/4A protease is a critical factor for hepatitis C virus (HCV) maturation that requires activation by NS4A. Synthetic peptide mutants of NS4A were found to inhibit NS3 function.
Abdelsattar M. Omar +7 more
doaj +1 more source

