Results 111 to 120 of about 8,749 (208)

Identification of new Trypanosoma cruzi-specific protein synthesis inhibitors by using a developed high-throughput in vitro translation assay. [PDF]

Int J Parasitol Drugs Drug Resist
Mantovani CC, Freitas FRN, Moraes CB, Dos Santos GRR, Cruz LR, Kratz JM, Aktas BH, Schenkman S.   +7 more
europepmc   +1 more source

Skeletal editing of anthranils via O-to-CN transmutation: access to ring-expanded quinazolines

A novel skeletal editing strategy of anthranils for the direct O-to-CN transmutation has been developed. This transformation enables the synthesis of ring-expanded quinazolines through three distinct approaches under metal-free conditions.
Saihui Song, Zicheng Liao, Shi Tang, Shuo-Wen Wang, Yongzhen Li, Lijuan Zhou, Jiajin Luo   +6 more
core   +1 more source

Discovery of cytotoxic indolo[1,2-<i>c</i>]quinazoline derivatives through scaffold-based design. [PDF]

Beilstein J Org Chem
Khabarov DV, Litvinova VA, Dezhenkova LG, Kaluzhny DN, Tikhomirov AS, Shchekotikhin AE.   +5 more
europepmc   +1 more source

Design, Synthesis, Antiproliferative Potency and In Silico Studies of Novel Alkynyl Quinazolines as Potential EGFR Inhibitors. [PDF]

Int J Mol Sci
Gkoutzivelaki A, Triantopoulou SI, Chiniadis L, Komiotis A, Triantis C, Komiotis D, Papakyriakou A, Pratsinis H, Manta S.   +8 more
europepmc   +1 more source

2-Azidobenzaldehyde-Enabled Construction of Quinazoline Derivatives: A Review. [PDF]

Int J Mol Sci
Qiu W, Zhan D, Ma X, Zhang X.
europepmc   +1 more source

Novel 5-Aryl-[1,2,4]triazoloquinazoline Fluorophores: Synthesis, Comparative Studies of the Optical Properties and ICT-Based Sensing Application. [PDF]

Molecules
Kopotilova AE, Permyakova JV, Starnovskaya ES, Moshkina TN, Novikov AS, Slepukhin PA, Nosova EV.   +6 more
europepmc   +1 more source

Multicomponent Synthesis of Multi-Target Quinazolines Modulating Cholinesterase, Oxidative Stress, and Amyloid Aggregation Activities for the Therapy of Alzheimer's Disease. [PDF]

Molecules
Chakhari S, Marco-Contelles J, Iriepa I, Carreiras MDC, Chabchoub F, Ismaili L, Refouvelet B.   +6 more
europepmc   +1 more source

Optimization of Quinazolines for Inhibition of <i>Trypanosoma brucei</i> Proliferation. [PDF]

ACS Med Chem Lett
Spijkers-Shaw S, Gadekar PK, Singh B, Kumar G, Sharma A, Hoffman B, Pollastri MP, Mensa-Wilmot K, Ferrins L.   +8 more
europepmc   +1 more source

Enhancing the MALDI-TOF MS Detection Mass Range of Saccharides Using a Reactive Composite Matrix. [PDF]

J Mass Spectrom
Wang S, Liu M, Ling L, Ding CF.
europepmc   +1 more source

A Tale of Two Cell Lines: Characterization of Differential Efficacy of Small Molecule Drugs Cediranib and NU-7441 on Primary Versus Metastatic Colorectal Cancer. [PDF]

Pharmacol Res Perspect
Tsang JD, Roberts CM.
europepmc   +1 more source