Results 11 to 20 of about 18,253 (267)
Application of Heteropoly Acids as Heterogeneous and Recyclable Catalysts for Friedländer Synthesis of Quinolines [PDF]
New convenient conditions for the Friedländer synthesis of quinolines are described. Quinolines were readily prepared in the presence of heteropolyacids as heterogeneous and recyclable catalysts in good yields.
Majid M. Heravi +4 more
doaj +2 more sources
Synthesis of two quinolines from one substrate: The beginning of regulating the duality of free radicals [PDF]
Poly-substituted quinolines are scaffolds with diverse applications as pharmaceuticals, agrochemicals, electroluminescent materials, and dyestuffs. Herein, we present an effective scheme for the green synthesis of two multiply substituted quinoline ...
Xuhong, Ren +8 more
core +1 more source
Multi-Substituted Quinolines as HIV-1 Integrase Allosteric Inhibitors
Allosteric HIV-1 integrase (IN) inhibitors, or ALLINIs, are a new class of antiviral agents that bind at the dimer interface of the IN, away from the enzymatic catalytic site and block viral replication by triggering an aberrant multimerization of the ...
Long Phi Dinh +7 more
doaj +1 more source
A series of fifteen silver (I) quinoline complexes Q1–Q15 have been synthesized and studied for their biological activities. Q1–Q15 were synthesized from the reactions of quinolinyl Schiff base derivatives L1–L5 (obtained by condensing 2 ...
Adesola A. Adeleke +6 more
doaj +1 more source
Chiral Phosphoric Acid Promoted Chiral 1H NMR Analysis of Atropisomeric Quinolines
An efficient enantioselective NMR analysis of atropisomeric quinolines in the promotion of chiral phosphoric acid is described, in which a variety of racemic 4-aryl quinolines were well-recognized with up to 0.17 ppm ΔΔδ value.
Junlin Wan, Jun Jiang, Juan Li
doaj +1 more source
An iron-catalyzed strategy for the rapid synthesis of indolo[2,3-c]quinolines has been developed. This cascade reaction involving alcohol oxidation, nitro reduction, and oxidative annulation was achieved in a one-pot.
Rong Li +6 more
doaj +1 more source
A convenient one-pot preparation of 2-methyl-3-(phenylthiomethyl)quinolines from Morita-Baylis-Hillman adducts via conjugate addition of thiols followed by reductive cyclization with Fe/AcOH was developed. The 2-methyl-3-(phenylthiomethyl)quinolines were
Ching-Fa Yao +4 more
doaj +1 more source
Iridium-catalyzed asymmetric transfer hydrogenation of quinolines with Hantzsch esters [PDF]
The iridium-catalyzed enantioselective transfer hydrogenation of quinolines with Hantzsch esters was developed with up to 88%, ee using [Ir(COD)Cl](2)/(S)-SegPhos/I-2 as a catalyst.
Zeng, Wei +3 more
core +1 more source
The pandemic that started in Wuhan (China) in 2019 has caused a large number of deaths, and infected people around the world due to the absence of effective therapy against coronavirus 2 of the severe acute respiratory syndrome (SARS-CoV-2).
Osvaldo Yañez +11 more
doaj +1 more source
Controlled partial transfer hydrogenation of quinolines by cobalt-amido cooperative catalysis
Controlling the partial reduction of quinolines is challenging, given the competing overreduction to tetrahydroquinolines. Here, the authors report a cobalt-amido cooperative catalyst for the selective, partial transfer hydrogenation of quinolines to 1,2-
Maofu Pang +5 more
doaj +1 more source

