Results 21 to 30 of about 19,883 (275)
A transition-metal-free method for the construction of 3-substituted or 3,4-disubstituted quinolines from readily available N,N-dimethyl enaminones and o-aminobenzyl alcohols is reported.
Kairui Rao +5 more
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Multi-Substituted Quinolines as HIV-1 Integrase Allosteric Inhibitors
Allosteric HIV-1 integrase (IN) inhibitors, or ALLINIs, are a new class of antiviral agents that bind at the dimer interface of the IN, away from the enzymatic catalytic site and block viral replication by triggering an aberrant multimerization of the ...
Long Phi Dinh +7 more
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Synthesis of two quinolines from one substrate: The beginning of regulating the duality of free radicals [PDF]
Poly-substituted quinolines are scaffolds with diverse applications as pharmaceuticals, agrochemicals, electroluminescent materials, and dyestuffs. Herein, we present an effective scheme for the green synthesis of two multiply substituted quinoline ...
Xuhong, Ren +8 more
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Diversely substituted quinolines via rhodium-catalyzed alkyne hydroacylation [PDF]
The Rh-catalyzed hydroacylative union of aldehydes and o-alkynyl anilines leads to 2-aminophenyl enones, and onwards to substituted quinolines. The mild reaction conditions employed in this chemistry result in a process that displays broad functional ...
Sarah M. Morrow (2561290) +3 more
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PERHALIDES OF QUINOLINE. [PDF]
n ...
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Newer Synthetic Approaches for the Disubstituted Quinolines from Aryl Amines [PDF]
Supervisor: Khan, Abu TalebThe thesis entitled “Newer Synthetic Approaches for the Disubstituted Quinolines from Aryl Amines” describes the synthesis of 2,3- and 2,4-disubstituted quinoline derivatives.
Ali, Saghir
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Efficient synthesis and antioxidation activities of ferrocenylpyrano-fused quinolines
Fifteen known ferrocenylpyrano-fused quinolines were synthesized efficiently via three-component Povarov reaction of 4-methyl-7-aminobenzopyranone, aromatic aldehydes, and ferrocenyl acetylene in the presence of cerium trifluoromethylsulfonate (Ce(OTf)3)
ZHANG Xiao-Ping +9 more
doaj
Quinolone and quinoline derivatives are frequently found as substructures in pharmaceutically active compounds. In this paper, we describe a procedure for the synthesis of azuleno[2,1-b]quinolones and quinolines from 2-arylaminoazulene derivatives, which
Taku Shoji +6 more
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N-(Quinolin-8-yl)quinoline-2-carboxamide [PDF]
In the title compound, C19H13N3O, the dihedral angle between the two quinoline systems is 11.54 (3)°. The molecular conformation is stabilized by intramolecular N—H...N and C—H...O hydrogen bonds, with N—H...N being bifurcated towards the two N atoms of the two quinoline rings.
Yanfeng Li, Hongbo Zhou, Xiaoping Shen
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Meta- or para-nitro-(pentafluorosulfonyl)benzenes underwent the Davis reaction with arylacetonitriles to provide the SF5-containing benzisoxazoles. Good yields were obtained with arylacetonitriles containing the electron-neutral or electron-donor group ...
Petr Beier, Tereza Pastýříková
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