Results 21 to 30 of about 414,318 (301)

Parallel solid-phase synthesis of diaryltriazoles

Beilstein Journal of Organic Chemistry, 2012
A series of substituted diaryltriazoles was prepared by a solid-phase-synthesis protocol using a modified Wang resin. The copper(I)- or ruthenium(II)-catalyzed 1,3-cycloaddition on the polymer bead allowed a rapid synthesis of the target compounds in a ...
Matthias Wrobel, Jeffrey Aubé, Burkhard König   +2 more
doaj   +1 more source

Solid-Phase Synthesis of a New Diphosphate 5-Aminoimidazole-4-carboxamide Riboside (AICAR) Derivative and Studies toward Cyclic AICAR Diphosphate Ribose

Molecules, 2011
The solid-phase synthesis of the first example of a new diphosphate AICAR derivative is reported. The new substance is characterized by the presence of a 5'-phosphate group while a second phosphate moiety is installed on a 5-hydroxypentyl chain attached ...
Gennaro Piccialli, Vincenzo Piccialli, Luciano Mayol, Michela Varra, Jussara Amato, Nicola Borbone, Giorgia Oliviero, Stefano D’Errico   +7 more
doaj   +1 more source

Photolabile Linkers for Solid-Phase Synthesis [PDF]

ACS Combinatorial Science, 2018
Photolabile linkers are the subjects of intense research because they allow the release of the target molecule simply by irradiation. Photochemical release of synthesis products is often facilitated without additional reagents under mild reaction conditions, which may even be environmentally friendly and appealing in the context of greener chemistry ...
Remi J. T. Mikkelsen, Katja E. Grier, Kim T. Mortensen, Thomas E. Nielsen, Katrine Qvortrup   +4 more
openaire   +5 more sources

Solid-Phase Synthesis of Substituted Tetramic Acids

, 2016
Solid-Phase Synthesis of Substituted Tetramic ...
Jay Matthews (3040941), Ralph A. Rivero (1993048)   +1 more
core   +2 more sources

New Solid Phase Synthesis of Distamycin Analogues

Molecules, 2011
A novel and straightforward solid phase synthesis of distamycin analogues containing benzene units has been developed.
Drozdowska Danuta
doaj   +1 more source

Rhodiasolv PolarClean – a greener alternative in solid-phase peptide synthesis

Green Chemistry Letters and Reviews, 2021
PolarClean, a green solvent prepared through the valorization of a byproduct of Nylon-66 manufacturing, shows an excellent capacity to dissolve all Fmoc-amino acids and key coupling reagents and additives.
Ashish Kumar, Anamika Sharma, Beatriz G. de la Torre, Fernando Albericio   +3 more
doaj   +1 more source

Solid-Phase Total Synthesis of Plusbacin A3

, 2022
The total synthesis of the depsipeptide natural product plusbacin A3 (1) utilizing solid-phase peptide synthesis (SPPS) was disclosed. A 3-hydroxy-proline derivative compatible with Fmoc SPPS was prepared by a diastereoselective Joullié–Ugi three ...
Toyotaka Sato, Satoshi Ichikawa, Motohiro Horiuchi, Satoshi Ichikawa (1310742), Shin-ichi Yokota, Kazuki Takashina, Akira Katsuyama (2796379), Satoshi Takahashi (77406), Kazuki Yamamoto, Rintaro Kaguchi (12249518), Toyotaka Sato (587317), Kazuki Takashina (12249515), Rintaro Kaguchi, Kazuki Yamamoto (1475920), Shin-ichi Yokota (587320), Motohiro Horiuchi (624763), Akira Katsuyama, Satoshi Takahashi   +17 more
core   +1 more source

Solid-Phase Synthesis of ?-Oligopeptides

CHIMIA, 1997
Fmoc-N-Protected ?-amino acids of (S)-configuration bearing the side chains of Ala, Val, Leu, and Phe in the 3- and 2-position have been prepared. Manual solid-phase synthesis (ortho-chlorotrityl-chloride resin) of the ?-heptapeptides H-?3-HVal-?
Gilles Guichard, Dieter Seebach
doaj   +2 more sources

Solid-Phase Unnatural Peptide Synthesis (UPS)

, 2016
Solid-Phase Unnatural Peptide Synthesis ...
Martin J. O'Donnell (2489491), William L. Scott (1314060), Changyou Zhou (2490022)   +2 more
core   +2 more sources

Optimized Solid Phase-Assisted Synthesis of Dendrons Applicable as Scaffolds for Radiolabeled Bioactive Multivalent Compounds Intended for Molecular Imaging

Molecules, 2014
Dendritic structures, being highly homogeneous and symmetric, represent ideal scaffolds for the multimerization of bioactive molecules and thus enable the synthesis of compounds of high valency which are e.g., applicable in radiolabeled form as ...
Gabriel Fischer, Björn Wängler, Carmen Wängler   +2 more
doaj   +1 more source