Journal of Enzyme Inhibition and Medicinal Chemistry, 2021 Sulphonamides and their isosteres are classical inhibitors of the carbonic anhydrase (CAs, EC 4.2.1.1) metalloenzymes. The protozoan pathogen Trichomonas vaginalis encodes two such enzymes belonging to the β-class, TvaCA1 and TvaCA2.
Linda J. Urbański +6 more
doaj +2 more sources
Investigation of sulphonamides effect on Anammox process
, 2010 The influence of selected sulphonamides such as sulphacetamide (SCM) and ptoluenesulphonamide(p-TSA) on the Anammox process was investigated. The short-term (14-hour) and long-term (90-day) exposure of mixed Anammox culture to SCM and p-TSA wasapplied ...
Medrzycka, K. +2 more
core +9 more sources
Antibacterial Effect of the In Vitro Interaction Between Clotrimazole and Chlorhexidine Against Staphylococcus pseudintermedius With Known Resistance Patterns Isolated From Canine Pyoderma. [PDF]
Vet Med SciThe 2:1 chlorhexidine–clotrimazole combination demonstrated enhanced antibacterial activity against canine Staphylococcus pseudintermedius isolates, including resistant strains. Reduced MIC values, predominantly additive interactions and absence of antagonism support its use as a promising topical strategy for canine pyoderma management.
Gallegos-Torres B +3 more
europepmc +2 more sources
The effect of sulphonamides on activated sludge dehydrogenase activity
, 2010 The effect of sulphonamides on activity of activated sludge dehydrogenase was studied. Three sulphonamides, such as sulphacetamide (SCM), sulphanilamide (SA), p-toluenesulphonamide(p-TSA), were selected for investigations and their concentrations ranged ...
Medrzycka, K. +2 more
core +9 more sources
Ultrasonicated synthesis of some potent antimicrobial aryl sulphonamides [PDF]
, 2021 1373-1377Nine N-(2,4-difluorophenyl) substituted benzene sulphonamides have been synthesized by ultrasonication method within short reaction time having more than 90% yield.
Thirunarayanan, G +5 more
core +3 more sources
Synthesis, characterization and anthelmintic activity evaluation of pyrimidine derivatives bearing carboxamide and sulphonamide moieties [PDF]
Journal of the Serbian Chemical Society, 2018 Pyrimidines, sulphonamides and carboxamides have shown a large number of pharmacological properties against different types of diseases including helminthiasis.
Ugwu David I. +2 more
doaj +1 more source
Halogen Bonding in Sulphonamide Co-Crystals: X···π Preferred over X···O/N?
Molecules, 2023 Sulphonamides have been one of the major pharmaceutical compound classes since their introduction in the 1930s. Co-crystallisation of sulphonamides with halogen bonding (XB) might lead to a new class of pharmaceutical-relevant co-crystals. We present the
Tobias Heinen +3 more
doaj +1 more source
Anaphylactic shock with intravenous furosemide: a rare undesired effect
MAMC Journal of Medical Sciences, 2020 Furosemide is a potent diuretic, with structural similarity to sulphonamide antibiotics. Its relative safety profile is one of the reasons to account for its widespread use.
Divya Gahlot +3 more
doaj +1 more source
Novel thiazolone-benzenesulphonamide inhibitors of human and bacterial carbonic anhydrases
Journal of Enzyme Inhibition and Medicinal Chemistry, 2023 A small library of novel thiazolone-benzenesulphonamides has been prepared and evaluated for their ability to inhibit three human cytosolic carbonic anhydrases (hCA I, hCA II, and hCA VII) and three bacterial carbonic anhydrases (MscCAβ, StCA1, and StCA2)
Morteza Abdoli +4 more
doaj +1 more source
, 2022 Archive of sulphonamides containing sub-folders named after each compound and its net charge. Every compound's folder contains a total of 20 files distributed into three sub-directories reporting QM (QM/), FF (FF/), and MD (MD ...
Giuliano Malloci (2060875) +5 more
core +1 more source